| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA678895 | B | Efficacy against human GABA-A receptor alpha-3-beta-3-gamma-2 subunits expressed in L(tk-) cells by whole-cell patch-clamp | Homo sapiens | 3 | ALA1149231 | cell-based format | Scientific Literature | |
| 2. | ALA678896 | B | Efficacy against human GABA-A receptor alpha-3-beta-3-gamma-2 subunits expressed in L(tk-) cells by whole-cell patch-clamp (No data) | Homo sapiens | 5 | ALA1149231 | cell-based format | Scientific Literature | |
| 3. | ALA678897 | B | Efficacy was determined against Gamma-aminobutyric acid A receptor, alpha 3 expressed in Xenopus oocytes | 15 | ALA1149231 | cell-based format | Scientific Literature | ||
| 4. | ALA678899 | B | In vitro binding affinity against Gamma-aminobutyric acid A receptor, alpha 3 expressed in L(tk) cells by displacement of [3H]Ro-151788 | 14 | ALA1149231 | cell-based format | Scientific Literature | ||
| 5. | ALA680327 | B | In vitro displacement of [3H]Ro-151788 from human GABA-A receptor alpha-3-beta-3-gamma-2 subunits expressed in L(tk-) cells | Homo sapiens | 1 | ALA1149231 | cell-based format | Scientific Literature | |
| 6. | ALA676772 | F | Agonistic activity against GABA-A receptor alpha-3-beta-3-gamma-2 | Homo sapiens | 1 | ALA1149126 | assay format | Scientific Literature | |
| 7. | ALA676773 | F | Inverse agonistic activity against GABA-A receptor alpha-3-beta-3-gamma-2 subunits | Homo sapiens | 2 | ALA1149126 | assay format | Scientific Literature | |
| 8. | ALA676774 | F | Partial agonistic activity against GABA-A receptor alpha-5-beta-3-gamma-2 | Homo sapiens | 1 | ALA1149126 | assay format | Scientific Literature | |
| 9. | ALA676775 | F | Partial agonistic activity against GABA-A receptor alpha-3-beta-3-gamma-2 subunits | Homo sapiens | 1 | ALA1149126 | assay format | Scientific Literature | |
| 10. | ALA676776 | F | Maximum percent change compared to GABA EC20 against GABA-A alpha-3-beta-3-gamma-2 receptor | Homo sapiens | 1 | ALA1149126 | assay format | Scientific Literature | |
| 11. | ALA676777 | F | Maximum percent change compared to GABA EC20 against GABA-A alpha-3-beta-3-gamma-2 receptor | Homo sapiens | 1 | ALA1149126 | assay format | Scientific Literature | |
| 12. | ALA676778 | F | Maximum percent change compared to GABA EC20 against GABA-A alpha-3-beta-3-gamma-2 receptor | Homo sapiens | 1 | ALA1149126 | assay format | Scientific Literature | |
| 13. | ALA676779 | F | Maximum percent change compared to GABA EC20 against GABA-A alpha-3-beta-3-gamma-2 receptor | Homo sapiens | 1 | ALA1149126 | assay format | Scientific Literature | |
| 14. | ALA678738 | F | Maximum percent change compared to GABA EC20 against GABA-A alpha-3-beta-3-gamma-2 receptor | Homo sapiens | 6 | ALA1149126 | assay format | Scientific Literature | |
| 15. | ALA678739 | F | Maximum percent change compared to GABA EC20 against GABA-A alpha-3-beta-3-gamma-2 receptor (not determined) | Homo sapiens | 1 | ALA1149126 | assay format | Scientific Literature | |
| 16. | ALA678741 | B | Binding affinity for human GABA-A receptor alpha-3-beta-3-gamma-2 subunits in L(tk-) cells | Homo sapiens | 62 | ALA1149126 | cell-based format | Scientific Literature | |
| 17. | ALA683025 | B | Percentage modulation of submaximal (EC20) response to GABA in Xenopus oocytes expressing human GABA-A alpha-3-beta-3-gamma-2 subunits | Homo sapiens | 12 | ALA1149152 | cell-based format | Scientific Literature | |
| 18. | ALA683026 | F | Percent change in electrophysiological response in Xenopus oocytes expressing Alpha3-beta3-gamma2 GABA-A receptor | 15 | ALA1148356 | cell-based format | Scientific Literature | ||
| 19. | ALA680428 | F | Percent change in electrophysiological response in Xenopus oocytes expressing alpha-3-beta-3-gamma-2 GABA-A receptor | Homo sapiens | 1 | ALA1148356 | cell-based format | Scientific Literature | |
| 20. | ALA680429 | F | Percent maximum change in electrophysiological response in Xenopus oocytes expressing alpha-3-beta-3-gamma-2 GABA-A receptor | Homo sapiens | 2 | ALA1148356 | cell-based format | Scientific Literature |
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