# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA749839 | B | Affinity for opiate receptors by measuring the inhibition of stereospecific binding of [3H]- naloxone in rat brain homogenates at a drug concentration of 2.0 x 10 E -5 M; Inactive | 1 | tissue-based format | Scientific Literature | |||
2. | ALA749840 | B | 50% Inhibition of stereospecific [3H]-naltrexone (10e-9 M) binding towards opiate receptor in rat brain homogenate | 7 | tissue-based format | Scientific Literature | |||
3. | ALA749841 | B | Ability to inhibit the specific binding of [3H]- dihydromorphine to opiate receptors in rat brain membrane preparation by 50% | 3 | cell membrane format | Scientific Literature | |||
4. | ALA749842 | B | Binding affinity against opiate receptor from rat neural membranes, using [3H]dihydromorphine as radioligand | 2 | assay format | Scientific Literature | |||
5. | ALA749843 | B | Concentration required to inhibit opiate receptor using radioligand [3H]- Etorphine | 6 | protein format | Scientific Literature | |||
6. | ALA749844 | B | Concentration required to inhibit opiate receptor using radioligand [3H]- Etorphine; Not tested | 1 | protein format | Scientific Literature | |||
7. | ALA749845 | B | Concentration required to inhibit stereospecific [3H]- naltrexone binding by 50% in rat brain homogenate | 5 | tissue-based format | Scientific Literature | |||
8. | ALA749846 | B | Inhibitory activity against opiate receptor in rat using [3H]naloxone as radioligand | 4 | assay format | Scientific Literature | |||
9. | ALA749847 | B | Inhibition of [3H]dihydromorphine binding to opiate receptor from rat neural membranes after incubation at 20 nM concentration at 37 degree C | 3 | cell membrane format | Scientific Literature | |||
10. | ALA753916 | B | Inhibition of [3H]naloxone binding to opiate receptor from rat neural membranes after incubation at 20 nM concentration at 37 degree C | 3 | cell membrane format | Scientific Literature | |||
11. | ALA858333 | B | Compound was evaluated for binding activity against [3H]sufentanil opiate receptor | Rattus norvegicus | 1 | protein format | Scientific Literature | ||
12. | ALA753917 | B | Ability to displace 50% of (+/-) ethylketocyclazocine (2.8) in rat brain homogenate | Rattus norvegicus | 1 | tissue-based format | Scientific Literature | ||
13. | ALA753918 | B | Ability to inhibit the specific binding of [3H]- dihydromorphine to opiate receptors in rat brain membrane preparation by 50% | Rattus norvegicus | 11 | cell membrane format | Scientific Literature | ||
14. | ALA753782 | B | Compound was evaluated for displacement of 8 nM [3H]dalamid from opioid receptor of rat brain membranes at the concentration of 0 moles | 2 | cell membrane format | Scientific Literature | |||
15. | ALA753783 | B | Compound was evaluated for displacement of 8 nM [3H]-Dalamid from opioid receptor of rat brain membranes at the concentration of 10e-10 moles | 2 | cell membrane format | Scientific Literature | |||
16. | ALA753784 | B | Compound was evaluated for displacement of 8 nM [3H]dalamid from opioid receptor of rat brain membranes at the concentration of 10e-4.2 moles | 2 | cell membrane format | Scientific Literature | |||
17. | ALA753785 | B | Compound was evaluated for displacement of 8 nM [3H]dalamid from opioid receptor of rat brain membranes at the concentration of 10e-4.6 moles | 2 | cell membrane format | Scientific Literature | |||
18. | ALA753921 | B | Compound was evaluated for displacement of 8 nM [3H]dalamid from opioid receptor of rat brain membranes at the concentration of 10e-5 moles | 2 | cell membrane format | Scientific Literature | |||
19. | ALA753922 | B | Compound was evaluated for displacement of 8 nM [3H]dalamid from opioid receptor of rat brain membranes at the concentration of 10e-5.2 moles | 2 | cell membrane format | Scientific Literature | |||
20. | ALA753923 | B | Compound was evaluated for displacement of 8 nM [3H]dalamid from opioid receptor of rat brain membranes at the concentration of 10e-5.6 moles | 2 | cell membrane format | Scientific Literature |