| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA656712 | F | Inhibitory concentration against 1 nM NPY induced [Ca2+] increase in CHO/dhFr- cells expressing recombinant human Y1 receptor; d=Not determined | 16 | cell-based format | Scientific Literature | |||
| 2. | ALA692301 | F | NPY Y1-antagonistic activity in HEL cells by measuring the inhibition of porcine NPY (10 nM) stimulated increase in the intracellular [Ca2+] concentration in a FURA-assay. | 29 | cell-based format | Scientific Literature | |||
| 3. | ALA752768 | F | Antagonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y1 receptors | 1 | assay format | Scientific Literature | |||
| 4. | ALA752769 | F | Antagonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y1 receptors | 3 | assay format | Scientific Literature | |||
| 5. | ALA752770 | B | Affinity for cloned Y1 receptor using [125I]PYY as radioligand | 4 | single protein format | Scientific Literature | |||
| 6. | ALA752771 | F | Antagonist potency for the inhibition of Forskolin stimulated cAMP synthesis in cells expressing cloned Y1 receptors | 2 | assay format | Scientific Literature | |||
| 7. | ALA752772 | B | Affinity for cloned Y1 receptor using [125I]PYY as radioligand | 5 | single protein format | Scientific Literature | |||
| 8. | ALA752773 | B | Selectivity ratio of Y1/Y2/Y4/Y5; 1/2/1/200 | 1 | single protein format | Scientific Literature | |||
| 9. | ALA752774 | B | Selectivity ratio of Y1/Y2/Y4/Y5; 1/50/110/150 | 1 | single protein format | Scientific Literature | |||
| 10. | ALA752775 | B | Selectivity ratio of Y1/Y2/Y4/Y5; 1/50/90/280 | 1 | single protein format | Scientific Literature | |||
| 11. | ALA752776 | B | Selectivity ratio of Y1/Y2/Y4/Y5; 1/790/3/1640 | 1 | single protein format | Scientific Literature | |||
| 12. | ALA748122 | B | Inhibitory activity tested against Human Neuropeptide Y1 Receptor. | 17 | single protein format | Scientific Literature | |||
| 13. | ALA755161 | B | Compound was tested for human Neuropeptide Y receptor type 1 | 1 | single protein format | Scientific Literature | |||
| 14. | ALA755162 | B | Compound was tested for its affinity to bind with Neuropeptide Y receptor type 1 | 5 | single protein format | Scientific Literature | |||
| 15. | ALA755163 | B | Affinity against Neuropeptide Y receptor Y1 in SK-N-MC cell line | 39 | cell-based format | Scientific Literature | |||
| 16. | ALA756250 | B | Binding affinity against Neuropeptide Y receptor type 1 using I-PYY as a radioligand in human neuroblastoma SK-N-MC cells | 1 | cell-based format | Scientific Literature | |||
| 17. | ALA756251 | B | Inhibition of I-PYY binding to Nueopeptide Y1 receptor expressed in human neuroblastoma SK-N-MC cells | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 18. | ALA756252 | B | Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]PYY | 22 | cell-based format | Scientific Literature | |||
| 19. | ALA756253 | B | Compound was evaluated for the inhibitory activity against human Neuropeptide Y receptor type 1 | 2 | single protein format | Scientific Literature | |||
| 20. | ALA756254 | B | Compound was evaluated for the inhibitory activity against human Neuropeptide Y receptor type 1; not tested | 1 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!