# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA655989 | Functional | Antagonistic effect on TPA-stimulated CD3 down-regulation in T-cells | 1 | ALA1126671 | assay format | Scientific Literature | ||
2. | ALA655990 | Functional | Antagonistic effect on TPA-stimulated CD3 down-regulation in T-cells | 1 | ALA1126671 | assay format | Scientific Literature | ||
3. | ALA822645 | Binding | Inhibition of protein kinase C(PKC), inhibition of phorbol binding by 80-100% at 38 uM | 2 | ALA1125489 | protein format | Scientific Literature | ||
4. | ALA860346 | Binding | Inhibition of PDBu activated protein kinase C at 1 nM | 1 | ALA1148572 | protein format | Scientific Literature | ||
5. | ALA860347 | Binding | Inhibition of PDBu activated protein kinase C at 100 nM | 1 | ALA1148572 | protein format | Scientific Literature | ||
6. | ALA860348 | Binding | Inhibition of PDBu activated protein kinase C at 10 uM | 1 | ALA1148572 | protein format | Scientific Literature | ||
7. | ALA770284 | Binding | Displacement of [3H]PDBu from Protein kinase C of CEM cells | Homo sapiens | 1 | ALA1126055 | cell-based format | Scientific Literature | |
8. | ALA770285 | Binding | Displacement of [3H]PDBu binding to Protein kinase C of CEM cells with 10% fetal calf serum | Homo sapiens | 1 | ALA1126055 | cell-based format | Scientific Literature | |
9. | ALA769343 | Binding | Binding to PKC in 3[H]-PBDU assay | 2 | ALA1126213 | protein format | Scientific Literature | ||
10. | ALA768501 | Binding | Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase C (not determined) | 1 | ALA1126493 | protein format | Scientific Literature | ||
11. | ALA768502 | Binding | Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase C | 3 | ALA1126493 | protein format | Scientific Literature | ||
12. | ALA768504 | Binding | Displacement of phorbol [3H]PDBu from protein kinase C; A - Did displace phorbol (PDBu) at 50 uM or less | 30 | ALA1149998 | protein format | Scientific Literature | ||
13. | ALA768505 | Binding | Displacement of phorbol [3H]PDBu from protein kinase C; Not tested | 26 | ALA1149998 | protein format | Scientific Literature |