#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA3721114	Binding	Inhibition of pyruvate dehydrogenase kinase (unknown origin) assessed as reduction in E1 phosphorylation incubated for 1 hr by DELFIA method	Homo sapiens	19	ALA3714766	protein format	Patent Bioactivity Data
2.	ALA3721115	Binding	Binding affinity to pyruvate dehydrogenase kinase (unknown origin) by VER-00160364 probe based fluorescence polarization assay	Homo sapiens	269	ALA3714766	assay format	Patent Bioactivity Data
3.	ALA3721116	Binding	Inhibition of pyruvate dehydrogenase kinase in human PC3 cells incubated for 90 mins by phospho(Ser293)E1alpha MSP ELISA method	Homo sapiens	30	ALA3714766	cell-based format	Patent Bioactivity Data
4.	ALA3734254	Binding	Inhibition of pyruvate dehydrogenase kinase in human PC3 cells incubated for 90 mins by phospho(Ser293)E1alpha MSP ELISA method	Homo sapiens	30	ALA3727364	cell-based format	Patent Bioactivity Data
5.	ALA767695	Functional	In vivo inhibion of pyruvate dehydrogenase kinase, increased oxidation of lactate	Homo sapiens	8	ALA1132309	organism-based format	Scientific Literature
6.	ALA767696	Binding	Inhibitory activity against Pyruvate dehydrogenase kinase	Sus scrofa	1	ALA1132309	protein format	Scientific Literature
7.	ALA767697	Binding	In vitro inhibitory activity against Pyruvate dehydrogenase kinase by primary enzymatic assay	Sus scrofa	18	ALA1132309	protein format	Scientific Literature
8.	ALA767698	Binding	Inhibitory activity against Pyruvate dehydrogenase kinase by primary enzymatic assay; inactive	Sus scrofa	2	ALA1132309	protein format	Scientific Literature
9.	ALA764813	Binding	In vitro inhibitory activity against pyruvate dehydrogenase kinase was determined		12	ALA1131823	protein format	Scientific Literature
10.	ALA764814	Binding	In vitro inhibitory activity against pyruvate dehydrogenase kinase was determined; Inactive at 1 mM concentration		12	ALA1131823	protein format	Scientific Literature
11.	ALA769458	Binding	Inhibition of porcine pyruvate dehydrogenase kinase (PDHK)in a primary enzymatic assay	Sus scrofa	90	ALA1133733	protein format	Scientific Literature
12.	ALA769459	Binding	In vitro inhibition of pyruvate dehydrogenase kinase (PDHK) in primary enzymatic assay; Inactive	Sus scrofa	2	ALA1133733	protein format	Scientific Literature
13.	ALA767850	Binding	In vitro inhibition of pyruvate dehydrogenase kinase (PDHK) in primary enzymatic assay; Inactive	Sus scrofa	9	ALA1133733	protein format	Scientific Literature
14.	ALA4311232	Binding	Inhibition of PDK in human NCI-H1975 cells assessed as reduction in phosphorylated S293 PDC E1 level at 10 uM by ELISA	Homo sapiens	4	ALA4308888	cell-based format	Scientific Literature
15.	ALA4311233	Binding	Inhibition of PDK in human NCI-H1975 cells assessed as reduction in phosphorylated S293 PDC E1 level by ELISA	Homo sapiens	2	ALA4308888	cell-based format	Scientific Literature
16.	ALA4311234	Binding	Inhibition of PDK in human NCI-H1975 cells assessed as reduction in phosphorylated S293 PDC E1 level by Western blot analysis	Homo sapiens	2	ALA4308888	cell-based format	Scientific Literature
17.	ALA4311241	Binding	Inhibition of PDK in human NCI-H1975 cells assessed as switch of pyruvate metabolism from lactate production to oxidative phosphorylation by measuring increase in ROS production at 1 to 10 uM measured after 4 hrs by DCFH-DA dye based assay	Homo sapiens	1	ALA4308888	cell-based format	Scientific Literature
18.	ALA4311242	Binding	Inhibition of PDK in human NCI-H1975 cells assessed as switch of pyruvate metabolism from lactate production to oxidative phosphorylation by measuring increase in oxygen consumption rate measured after 2 hrs	Homo sapiens	1	ALA4308888	cell-based format	Scientific Literature
19.	ALA4311243	Binding	Inhibition of PDK in human NCI-H1975 cells assessed as switch of pyruvate metabolism from lactate production to oxidative phosphorylation by measuring decrease in lactate production at 1 to 10 uM measured after 4 hrs	Homo sapiens	1	ALA4308888	cell-based format	Scientific Literature
20.	ALA4369509	Binding	Inhibition of PDK in human NCI-H1975 cells assessed as reduction in PDC phosphorylation at 2 uM measured after 12 hrs under hypoxic condition by Western blot analysis	Homo sapiens	3	ALA4368877	cell-based format	Scientific Literature