| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA699616 | F | Inhibition against GRO-alpha driven human neutrophil chemotaxis | 23 | ALA1135131 | assay format | Scientific Literature | ||
| 2. | ALA696549 | B | Compound was tested for inhibitory activity against Interleukin-8 receptor | 1 | ALA1150989 | protein format | Scientific Literature | ||
| 3. | ALA696550 | B | Inhibitory activity against interleukin-8 receptor using [125I]IL8 | 37 | ALA1150989 | protein format | Scientific Literature | ||
| 4. | ALA850062 | B | Inhibition ratio of CXCR 2 receptor to that of CXCR 1 receptor | Homo sapiens | 8 | ALA1149089 | protein format | Scientific Literature | |
| 5. | ALA833397 | F | Inhibition of CXCL8-induced chemotaxis in human polymorphonuclear cells | Homo sapiens | 8 | ALA1145151 | assay format | Scientific Literature | |
| 6. | ALA826538 | F | Inhibition of CXCL8-induced chemotaxis of human polymorphonuclear cells at 10e-8 M | Homo sapiens | 74 | ALA1145151 | assay format | Scientific Literature | |
| 7. | ALA826659 | F | Inhibition of interleukin-8 induced chemotaxis of human polymorphonuclear cells at 100 nM | Homo sapiens | 10 | ALA1145151 | assay format | Scientific Literature | |
| 8. | ALA877356 | F | Inhibition of CXCL8-induced chemotaxis of human polymorphonuclear cells at 10e-6 M: not active | Homo sapiens | 1 | ALA1145151 | assay format | Scientific Literature | |
| 9. | ALA877357 | F | Inhibition of CXCL8-induced chemotaxis of human polymorphonuclear cells at 10e-8 M: not active | Homo sapiens | 32 | ALA1145151 | assay format | Scientific Literature | |
| 10. | ALA862383 | F | Inhibition of GROalpha-stimulated intracellular calcium mobilisation in human neutrophils by FLIPR | Homo sapiens | 2 | ALA1149469 | cell-based format | Scientific Literature | |
| 11. | ALA912818 | B | Selectivity for CXCR2 over CXCR1 | Homo sapiens | 1 | ALA1138214 | protein format | Scientific Literature | |
| 12. | ALA912819 | F | Inhibition of CXCL8-induced human neutrophil chemotaxis | Homo sapiens | 3 | ALA1138214 | assay format | Scientific Literature | |
| 13. | ALA908415 | B | Selectivity for CXCR2 over CXCR1 | Homo sapiens | 1 | ALA1139694 | protein format | Scientific Literature | |
| 14. | ALA896520 | B | Ratio of IC50 for CXCR2 receptor to IC50 CXCR1 receptor | Homo sapiens | 7 | ALA1149534 | protein format | Scientific Literature | |
| 15. | ALA927479 | F | Antagonist activity at CXCR1/CXCR2 in human PMN cells assessed as inhibition of IL8-mediated myeloperoxidase release | Homo sapiens | 14 | ALA1140777 | cell-based format | Scientific Literature | |
| 16. | ALA927480 | F | Antagonist activity at CXCR1/CXCR2 in human PMN cells assessed as inhibition of GROalpha-mediated myeloperoxidase release | Homo sapiens | 9 | ALA1140777 | cell-based format | Scientific Literature | |
| 17. | ALA927482 | F | Antagonist activity at CXCR1/CXCR2 in human PMN cells assessed as inhibition of GROalpha-mediated myeloperoxidase release at 1 uM | Homo sapiens | 5 | ALA1140777 | cell-based format | Scientific Literature | |
| 18. | ALA1003796 | B | Displacement of [125I]IL8 from human CXCR1/2 expressed in CHO cells at 10 uM | Homo sapiens | 1 | ALA1139391 | cell-based format | Scientific Literature | |
| 19. | ALA2026802 | B | Inhibition of CXCR1/2 in human polymorphonucleate cells assessed as inhibition of CXCL8-induced chemotaxis at 10'-8 M incubated for 15 mins prior to CXCL8-induction measured after 45 mins | Homo sapiens | 22 | ALA2021812 | assay format | Scientific Literature | |
| 20. | ALA3386571 | F | Antagonist activity at CXCR1/CXCR2 in human PMNs assessed as inhibition of CXCL8-induced intracellular Ca2+ release by fluorescence based calcium flux assay | Homo sapiens | 1 | ALA3352272 | cell-based format | Scientific Literature |
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