| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA859561 | B | Displacement of [125I-Tyr10] from halphaCGRP expressed in human neuroblastoma SK-N-MC cells | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 2. | ALA859562 | B | Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cells | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 3. | ALA858539 | F | Antagonist activity on halphaCGRP-induced cAMP accumulation at human neuroblastoma SK-N-MC cells | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 4. | ALA866916 | B | Displacement of [125I]CGRP from human cloned CLR/RAMP1 receptor expressed in E10 cells | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 5. | ALA866917 | B | Displacement of [125I]CGRP from human cloned CLR/RAMP1 receptor expressed in SK-N-MC cells at 100 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA864503 | F | Antagonist activity at human cloned CLR/RAMP1 receptor expressed in E10 cells measured as inhibition of CGRP-mediated cAMP production | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 7. | ALA865680 | F | Antagonist activity at human cloned CLR/RAMP1 receptor expressed in E10 cells measured as inhibition of CGRP-mediated cAMP production at 17 uM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA2040005 | B | Displacement of [125I]CGRP from human recombinant CALCRL/RAMP1 receptor expressed in HEK293 cells after 3 hrs | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 9. | ALA897783 | B | Displacement of [125I]CGRP from human CL receptor in RAMP1 membranes | Homo sapiens | 17 | cell membrane format | Scientific Literature | ||
| 10. | ALA897784 | F | Antagonist activity at human CGRP receptor in E10 cells assessed as inhibition of cAMP production | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 11. | ALA897787 | B | Displacement of [125I]CGRP from human CL receptor in RAMP1 membranes at 100 uM | Homo sapiens | 2 | cell membrane format | Scientific Literature | ||
| 12. | ALA3102085 | B | Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranes | Homo sapiens | 27 | cell-based format | Scientific Literature | ||
| 13. | ALA3881288 | B | Displacement of [125I]hCGRP from human recombinant CGRP receptor expressed in HEK293 cell membranes incubated for 3 hrs by scintillation counting method | Homo sapiens | 16 | cell-based format | Patent Bioactivity Data | ||
| 14. | ALA4612974 | B | Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintillation counting method | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 15. | ALA4612975 | F | Antagonist activity at human CGRP receptor in human SK-N-MC cells assessed as inhibition of CGRP-induced cAMP production preincubated for 30 mins followed by CGRP addition and measured after 30 mins by HTRF assay | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 16. | ALA4617610 | B | Inhibition of human CLR/RAMP1 | Homo sapiens | 19 | protein complex format | Scientific Literature | ||
| 17. | ALA4617617 | B | Antagonist activity at human CLR/RAMP1 | Homo sapiens | 2 | protein complex format | Scientific Literature | ||
| 18. | ALA4617619 | F | Inhibition of human CLR/RAMP1 by cAMP assay | Homo sapiens | 2 | protein complex format | Scientific Literature | ||
| 19. | ALA4880124 | B | CGRP (h) CEREP ligand profiling | Homo sapiens | 1 | protein complex format | Donated Chemical Probes - SGC Frankfurt | ||
| 20. | ALA4880173 | B | CGRP (h) Ligand binding assay | Homo sapiens | 1 | protein complex format | Donated Chemical Probes - SGC Frankfurt |
The page will load shortly, Thanks for your patience!