# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA859561 | B | Displacement of [125I-Tyr10] from halphaCGRP expressed in human neuroblastoma SK-N-MC cells | Homo sapiens | 3 | ALA1147739 | cell-based format | Scientific Literature | |
2. | ALA859562 | B | Displacement of [3H-propionyl-K24] from halphaCGRP expressed in human neuroblastoma SK-N-MC cells | Homo sapiens | 14 | ALA1147739 | cell-based format | Scientific Literature | |
3. | ALA858539 | F | Antagonist activity on halphaCGRP-induced cAMP accumulation at human neuroblastoma SK-N-MC cells | Homo sapiens | 4 | ALA1147739 | cell-based format | Scientific Literature | |
4. | ALA866916 | B | Displacement of [125I]CGRP from human cloned CLR/RAMP1 receptor expressed in E10 cells | Homo sapiens | 11 | ALA1147686 | cell-based format | Scientific Literature | |
5. | ALA866917 | B | Displacement of [125I]CGRP from human cloned CLR/RAMP1 receptor expressed in SK-N-MC cells at 100 uM | Homo sapiens | 1 | ALA1147686 | cell-based format | Scientific Literature | |
6. | ALA864503 | F | Antagonist activity at human cloned CLR/RAMP1 receptor expressed in E10 cells measured as inhibition of CGRP-mediated cAMP production | Homo sapiens | 9 | ALA1147686 | cell-based format | Scientific Literature | |
7. | ALA865680 | F | Antagonist activity at human cloned CLR/RAMP1 receptor expressed in E10 cells measured as inhibition of CGRP-mediated cAMP production at 17 uM | Homo sapiens | 1 | ALA1147686 | cell-based format | Scientific Literature | |
8. | ALA897783 | B | Displacement of [125I]CGRP from human CL receptor in RAMP1 membranes | Homo sapiens | 17 | ALA1149654 | cell membrane format | Scientific Literature | |
9. | ALA897784 | F | Antagonist activity at human CGRP receptor in E10 cells assessed as inhibition of cAMP production | Homo sapiens | 14 | ALA1149654 | cell-based format | Scientific Literature | |
10. | ALA897787 | B | Displacement of [125I]CGRP from human CL receptor in RAMP1 membranes at 100 uM | Homo sapiens | 2 | ALA1149654 | cell membrane format | Scientific Literature | |
11. | ALA2040005 | B | Displacement of [125I]CGRP from human recombinant CALCRL/RAMP1 receptor expressed in HEK293 cells after 3 hrs | Homo sapiens | 7 | ALA2034981 | cell-based format | Scientific Literature | |
12. | ALA3102085 | B | Displacement of [125I]-hCGRP from human CALCRL/RAMP1 expressed in HEK293 cell membranes | Homo sapiens | 27 | ALA3098057 | cell-based format | Scientific Literature | |
13. | ALA3881288 | B | Displacement of [125I]hCGRP from human recombinant CGRP receptor expressed in HEK293 cell membranes incubated for 3 hrs by scintillation counting method | Homo sapiens | 16 | ALA3880433 | cell-based format | Patent Bioactivity Data | |
14. | ALA4612974 | B | Displacement of [3H]telcagepant from recombinant human CLR/RAMP1 expressed in Sf21 insect cell membranes measured after 60 mins by microbeta scintillation counting method | Homo sapiens | 9 | ALA4610123 | cell-based format | Scientific Literature | |
15. | ALA4612975 | F | Antagonist activity at human CGRP receptor in human SK-N-MC cells assessed as inhibition of CGRP-induced cAMP production preincubated for 30 mins followed by CGRP addition and measured after 30 mins by HTRF assay | Homo sapiens | 9 | ALA4610123 | cell-based format | Scientific Literature | |
16. | ALA4617610 | B | Inhibition of human CLR/RAMP1 | Homo sapiens | 19 | ALA4616627 | protein complex format | Scientific Literature | |
17. | ALA4617617 | B | Antagonist activity at human CLR/RAMP1 | Homo sapiens | 2 | ALA4616627 | protein complex format | Scientific Literature | |
18. | ALA4617619 | F | Inhibition of human CLR/RAMP1 by cAMP assay | Homo sapiens | 2 | ALA4616627 | protein complex format | Scientific Literature | |
19. | ALA4880124 | B | CGRP (h) CEREP ligand profiling | Homo sapiens | 1 | ALA4507256 | protein complex format | Donated Chemical Probes - SGC Frankfurt | |
20. | ALA4880173 | B | CGRP (h) Ligand binding assay | Homo sapiens | 1 | ALA4507257 | protein complex format | Donated Chemical Probes - SGC Frankfurt |