| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA869928 | F | Inhibition of agonist site of GABAA receptor at 1 nM | 1 | ALA1148572 | assay format | Scientific Literature | ||
| 2. | ALA853023 | F | Inhibition of agonist site of GABAA receptor at 100 nM | 1 | ALA1148572 | assay format | Scientific Literature | ||
| 3. | ALA852986 | F | Inhibition of agonist site of GABAA receptor at 10 uM | 1 | ALA1148572 | assay format | Scientific Literature | ||
| 4. | ALA964519 | F | Agonist activity at human alpha-1-beta-2-gamma-2L GABAA receptor expressed in Xenopus oocytes assessed as inhibition of current production by two electrode voltage clamp method | Homo sapiens | 6 | ALA1157459 | cell-based format | Scientific Literature | |
| 5. | ALA964520 | F | Antagonist activity at human alpha-1-beta-2-gamma-2L GABAA receptor expressed in Xenopus oocytes assessed as inhibition of current production by two electrode voltage clamp method | Homo sapiens | 1 | ALA1157459 | cell-based format | Scientific Literature | |
| 6. | ALA964521 | B | Activity at human alpha-1-beta-2-gamma-2L GABAA receptor expressed in Xenopus oocytes assessed as inhibition of current production at 600 uM by two electrode voltage clamp method relative to GABA | Homo sapiens | 9 | ALA1157459 | cell-based format | Scientific Literature | |
| 7. | ALA1047262 | B | Binding affinity to human GABAA receptor | Homo sapiens | 1 | ALA1156026 | protein complex format | Scientific Literature | |
| 8. | ALA1117107 | F | Partial agonist activity at human alpha-1-beta-3-gamma-2 GABAA receptor expressed in Lkt cells | Homo sapiens | 1 | ALA1156265 | cell-based format | Scientific Literature | |
| 9. | ALA1120210 | F | Partial agonist activity at human GABAA receptor | Homo sapiens | 1 | ALA1158602 | assay format | Scientific Literature | |
| 10. | ALA1120211 | F | Partial agonist activity at human GABAA receptor at 3 uM | Homo sapiens | 1 | ALA1158602 | assay format | Scientific Literature | |
| 11. | ALA1247887 | B | Binding affinity to human recombinant GABAA receptor | Homo sapiens | 1 | ALA1240532 | protein complex format | Scientific Literature | |
| 12. | ALA1259912 | B | Binding affinity to human GABAA receptor | Homo sapiens | 3 | ALA1255169 | protein complex format | Scientific Literature | |
| 13. | ALA2169245 | F | Agonist activity at human alpha1beta2gamma2L GABAA receptor expressed in Xenopus oocytes assessed as potentiation of channel current response by two-electrode voltage clamp electrophysiology assay relative to control | Homo sapiens | 2 | ALA2163281 | cell-based format | Scientific Literature | |
| 14. | ALA2169246 | F | Agonist activity at human alpha1beta2gamma2L GABAA receptor expressed in Xenopus oocytes assessed as potentiation of GABA-induced current response at 4.4 uM by two-electrode voltage clamp electrophysiology assay relative to control | Homo sapiens | 1 | ALA2163281 | cell-based format | Scientific Literature | |
| 15. | ALA2169247 | F | Agonist activity at human alpha1beta2gamma2L GABAA receptor expressed in Xenopus oocytes assessed as potentiation of GABA-induced current response at 6 uM by two-electrode voltage clamp electrophysiology assay relative to control | Homo sapiens | 1 | ALA2163281 | cell-based format | Scientific Literature | |
| 16. | ALA2169248 | F | Agonist activity at human alpha1beta2gamma2L GABAA receptor expressed in Xenopus oocytes assessed as potentiation of channel current response by two-electrode voltage clamp electrophysiology assay | Homo sapiens | 3 | ALA2163281 | cell-based format | Scientific Literature | |
| 17. | ALA2169249 | F | Agonist activity at human alpha1beta2gamma2L GABAA receptor expressed in Xenopus oocytes assessed as potentiation of GABA-induced current response at 30 to 100 uM by two-electrode voltage clamp electrophysiology assay relative to control | Homo sapiens | 1 | ALA2163281 | cell-based format | Scientific Literature | |
| 18. | ALA2169250 | F | Agonist activity at human alpha1beta2gamma2L GABAA receptor expressed in Xenopus oocytes assessed as potentiation of GABA-induced current response at 100 uM by two-electrode voltage clamp electrophysiology assay relative to control | Homo sapiens | 1 | ALA2163281 | cell-based format | Scientific Literature | |
| 19. | ALA2169251 | F | Agonist activity at human alpha1beta2gamma2L GABAA receptor expressed in Xenopus oocytes assessed as potentiation of GABA-induced current response by two-electrode voltage clamp electrophysiology assay | Homo sapiens | 2 | ALA2163281 | cell-based format | Scientific Literature | |
| 20. | ALA3054658 | B | Displacement of [3H]TBOB from GABAA receptor (unknown origin) at 10 uM | Homo sapiens | 6 | ALA3046958 | protein complex format | Scientific Literature |
The page will load shortly, Thanks for your patience!