| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA681840 | B | Binding affinity for human GABA-A receptor alpha-2-beta-2-gamma-2 expressed in L(tk-) cell membranes | Homo sapiens | 11 | ALA1129572 | cell-based format | Scientific Literature | |
| 2. | ALA824292 | F | Potentiation of GABA-evoked Cl- currents in Xenopus oocytes expressing human alpha-2-beta-2-gamma-2 subunits | Homo sapiens | 3 | ALA1130157 | cell-based format | Scientific Literature | |
| 3. | ALA824293 | F | Maximal potentiation of GABA-evoked Cl- currents in Xenopus oocytes expressing human alpha-2-beta-2-gamma-2 subunits | Homo sapiens | 3 | ALA1130157 | cell-based format | Scientific Literature | |
| 4. | ALA831818 | B | Effective concentration against GABA-evoked chloride currents mediated by human Gamma-aminobutyric acid GABA-A receptor alpha2-beta2-gamma2L expressed in Xenopus oocytes | Homo sapiens | 26 | ALA1145214 | cell-based format | Scientific Literature | |
| 5. | ALA832867 | B | Effective concentration against GABA-evoked chloride currents mediated by human Gamma-aminobutyric acid GABA-A receptor alpha2-beta2-gamma2L expressed in Xenopus oocytes; ND = not determinable | Homo sapiens | 3 | ALA1145214 | cell-based format | Scientific Literature | |
| 6. | ALA829858 | B | Maximal efficacy for GABA-evoked chloride currents mediated by human Gamma-aminobutyric acid GABA-A receptor alpha2-beta2-gamma2L expressed in Xenopus oocytes | Homo sapiens | 29 | ALA1145214 | cell-based format | Scientific Literature | |
| 7. | ALA898324 | B | Displacement of [3H]EBOB from human recombinant GABA alpha-1-beta-2-gamma-2 receptor expressed in HEK293 cells | Homo sapiens | 37 | ALA1149606 | cell-based format | Scientific Literature | |
| 8. | ALA924987 | B | Binding affinity to GABA alpha-2-beta-2-gamma-2 receptor | Homo sapiens | 1 | ALA1140697 | protein complex format | Scientific Literature | |
| 9. | ALA942241 | B | Displacement of [3H]Ro-151788 from benzodiazepine binding site of GABAA alpha-2-beta-2-gamma-2 receptor expressed in HEK293T cells | 4 | ALA1152298 | cell-based format | Scientific Literature | ||
| 10. | ALA1065532 | B | Displacement of [3H]flunitrezepam from GABA-A alpha-2-beta-2-gamma-2 receptor by liquid scintillation counting | 1 | ALA1157703 | protein complex format | Scientific Literature | ||
| 11. | ALA1282596 | B | Binding affinity to human recombinant GABA alpha-2-beta-2-gamma-2 receptor | Homo sapiens | 1 | ALA1275264 | protein complex format | Scientific Literature | |
| 12. | ALA2173575 | B | Displacement of [3H]flumazenil from human recombinant GABA-A alpha2beta2gamma2L receptor expressed in HEK293 cells | Homo sapiens | 2 | ALA2169854 | cell-based format | Scientific Literature | |
| 13. | ALA2317986 | B | Agonist activity at human GABAA alpha2beta2gamma2S receptor expressed in TSA201 cells after 1 min by FLIPR assay relative to GABA | Homo sapiens | 1 | ALA2311400 | cell-based format | Scientific Literature | |
| 14. | ALA2318266 | B | Agonist activity at human GABAA alpha2beta2gamma2S receptor expressed in TSA201 cells after 1 min by FLIPR assay | Homo sapiens | 3 | ALA2311400 | cell-based format | Scientific Literature | |
| 15. | ALA2353551 | B | Displacement of [3H]Ro15-1788 from recombinant GABA-A alpha2beta2gamma2 receptor benzodiazepine binding site (unknown origin) at 10 uM after 1 hr relative to control | Homo sapiens | 2 | ALA2346497 | protein complex format | Scientific Literature | |
| 16. | ALA3116676 | B | Modulation of GABAA alpha2beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of EC3 to 10 GABA-induced chloride ion current at holding potential -70 mV at 1 to 300 uM by two-microelectrode voltage clamp assay relative to GABA-treated control | Homo sapiens | 1 | ALA3112517 | cell-based format | Scientific Literature | |
| 17. | ALA3116682 | B | Modulation of GABAA alpha2beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of EC3 to 10 GABA-induced chloride ion current at holding potential -70 mV by two-microelectrode voltage clamp assay | Homo sapiens | 1 | ALA3112517 | cell-based format | Scientific Literature | |
| 18. | ALA3297503 | B | Modulation of GABAA alpha2beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as modulation of GABA-induced maximal chloride ion current at holding potential -70 mV by two-microelectrode voltage clamp assay relative to GABA-treated control | Homo sapiens | 2 | ALA3286229 | cell-based format | Scientific Literature | |
| 19. | ALA3297509 | B | Modulation of GABAA alpha2beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as modulation of GABA-induced chloride ion current at holding potential -70 mV by two-microelectrode voltage clamp assay | Homo sapiens | 2 | ALA3286229 | cell-based format | Scientific Literature | |
| 20. | ALA3370257 | B | Agonist activity at human GABAAalpha2beta2gamma2S receptor expressed in tsA-201cells by FLIPR membrane potential blue assay | Homo sapiens | 6 | ALA3351648 | cell membrane format | Scientific Literature |
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