| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA661783 | B | Inhibition of ligand-stimulated autophosphorylation of EGFR/HER2 chimeric receptor expressed in NIH3T3 cells | 11 | ALA1130506 | cell-based format | Scientific Literature | ||
| 2. | ALA677877 | B | Concentration needed to inhibit the autophosphorylation of the cytoplasmic domain of Epidermal growth factor receptor using DELFIA/time-resolved fluorimetry. | 51 | ALA1133627 | protein format | Scientific Literature | ||
| 3. | ALA689286 | F | Inhibitory concentration against ErbB2/neu (HER-2) by autophosphorylation | 25 | ALA1126897 | assay format | Scientific Literature | ||
| 4. | ALA689287 | F | Inhibition of ErbB2/neu (HER-2) autophosphorylation (Not determined) | Homo sapiens | 2 | ALA1126897 | assay format | Scientific Literature | |
| 5. | ALA689293 | B | Inhibition of human HER-2 | Homo sapiens | 4 | ALA1147483 | protein format | Scientific Literature | |
| 6. | ALA702407 | F | In vitro efficacy (average) against HN5 (EGFR) and BT474 (erbB2) tumor cell proliferation | Homo sapiens | 1 | ALA1146682 | assay format | Scientific Literature | |
| 7. | ALA815615 | F | Inhibition of EGFR and erbB2 overexpressing tumor cell proliferation | Homo sapiens | 6 | ALA1136583 | assay format | Scientific Literature | |
| 8. | ALA846175 | B | Inhibition of EGFR and ErbB-2 average ratio | 6 | ALA1136583 | protein format | Scientific Literature | ||
| 9. | ALA845349 | F | Selective inhibition of EGFR/erbB2 tumor cell proliferation over normal HFF cells | Homo sapiens | 6 | ALA1136583 | cell-based format | Scientific Literature | |
| 10. | ALA880405 | B | Selectivity for EGF receptor and erbB2 | 1 | ALA1134080 | protein format | Scientific Literature | ||
| 11. | ALA848965 | B | Selectivity for EGF receptor and c-erbB-2 | 9 | ALA1134080 | protein format | Scientific Literature | ||
| 12. | ALA873337 | F | Inhibition of EGF-stimulated human umbilical vein endothelial cell proliferation | Homo sapiens | 7 | ALA1138664 | cell-based format | Scientific Literature | |
| 13. | ALA835868 | F | Inhibition of EGF-stimulated human umbilical vein endothelial cell proliferation; ND= not determined | Homo sapiens | 2 | ALA1138664 | cell-based format | Scientific Literature | |
| 14. | ALA887680 | B | Selectivity for erbB2 over EGFR | Homo sapiens | 45 | ALA1144645 | protein format | Scientific Literature | |
| 15. | ALA1060286 | B | Inhibition of HER1/HER2 phosphorylation in human N87 cells by Western blot | Homo sapiens | 1 | ALA1154610 | cell-based format | Scientific Literature | |
| 16. | ALA1060287 | B | Inhibition of HER1/HER2-mediated AKT phosphorylation in human GEO cells by Western blot | Homo sapiens | 1 | ALA1154610 | cell-based format | Scientific Literature | |
| 17. | ALA1060288 | B | Inhibition of HER1/HER2-mediated MAPK phosphorylation in human GEO cells by Western blot | Homo sapiens | 1 | ALA1154610 | cell-based format | Scientific Literature | |
| 18. | ALA1060289 | B | Inhibition of epidermal growth factor-induced HER1/HER2 heterodimer formation in human AU565 cells at 1 uM by immunoprecipitation | Homo sapiens | 1 | ALA1154610 | cell-based format | Scientific Literature | |
| 19. | ALA4816058 | B | Inhibition of HER2/EGFR dimerization in human A549 cells incubated for 48 hrs by proximity ligation assay | Homo sapiens | 1 | ALA4813972 | cell-based format | Scientific Literature | |
| 20. | ALA4816060 | B | Inhibition of HER2/EGFR dimerization in human Calu-3 cells incubated for 48 hrs by proximity ligation assay | Homo sapiens | 1 | ALA4813972 | cell-based format | Scientific Literature |
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