| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA680339 | B | Inhibition of [3H]CGP-27492 binding to cat Gamma-aminobutyric acid type B receptor | Felis catus | 2 | ALA1128747 | protein complex format | Scientific Literature | |
| 2. | ALA682870 | B | Inhibition of [3H]baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellum | Felis catus | 3 | ALA1128747 | tissue-based format | Scientific Literature | |
| 3. | ALA682871 | B | Inhibition of [3H]-baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellum | Felis catus | 14 | ALA1128747 | tissue-based format | Scientific Literature | |
| 4. | ALA682872 | B | Inhibition of [3H]baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellum at 10e-5 M | Felis catus | 1 | ALA1128747 | tissue-based format | Scientific Literature | |
| 5. | ALA682873 | B | Inhibition of [3H]baclofen binding to Gamma-aminobutyric acid type B receptor of cat cerebellum at 10e-5 M | Felis catus | 3 | ALA1128747 | tissue-based format | Scientific Literature | |
| 6. | ALA682874 | B | Inhibition of Gamma-aminobutyric acid type B receptor | Bos taurus | 2 | ALA1128116 | protein complex format | Scientific Literature | |
| 7. | ALA682875 | F | Antagonistic potency against Gamma-aminobutyric acid type B receptor of guinea pig ileum | Cavia porcellus | 1 | ALA1136325 | tissue-based format | Scientific Literature | |
| 8. | ALA682876 | F | Antagonistic potency against Gamma-aminobutyric acid type B receptor in guinea pig ileum, inactive up to 100 uM | Cavia porcellus | 2 | ALA1136325 | tissue-based format | Scientific Literature | |
| 9. | ALA679658 | B | Inhibition of mammalian Gamma-aminobutyric acid type B receptor (Inactive) | 1 | ALA1150031 | protein complex format | Scientific Literature | ||
| 10. | ALA679659 | F | Inhibition of mammalian Gamma-aminobutyric acid type B receptor (potent agonist) | 1 | ALA1150031 | assay format | Scientific Literature | ||
| 11. | ALA881980 | B | Percent inhibition against GABA-B receptor at 1 uM | 3 | ALA1140374 | protein complex format | Scientific Literature | ||
| 12. | ALA899070 | F | Activity at GABAB 1b/2 receptor expressed in CHO-K1 cells assessed as effect on glutamate-induced [35S]GTP-gamma-S binding at 2.5 uM | Homo sapiens | 38 | ALA1137529 | cell-based format | Scientific Literature | |
| 13. | ALA899071 | F | Activity at GABAB 1b/2 receptor expressed in CHO-K1 cells assessed as effect on glutamate-induced [35S]GTP-gamma-S binding at 25 uM | Homo sapiens | 38 | ALA1137529 | cell-based format | Scientific Literature | |
| 14. | ALA899072 | F | Activity at GABAB 1b/2 receptor expressed in CHO-K1 cells assessed as effect on glutamate-induced [35S]GTP-gamma-S binding | Homo sapiens | 11 | ALA1137529 | cell-based format | Scientific Literature | |
| 15. | ALA899073 | F | Activity at GABAB 1b/2 receptor expressed in CHO-K1 cells assessed as effect on glutamate-induced [35S]GTP-gamma-S binding in presence of 1 uM GABA | Homo sapiens | 11 | ALA1137529 | cell-based format | Scientific Literature | |
| 16. | ALA1679957 | F | Antagonist activity at human recombinant GABAb 1b/2 receptor expressed in Xenopus laevis oocytes co-expressing GIRK1/4 assessed as inhibition of GABA-induced current by two electrode voltage clamp technique | Homo sapiens | 2 | ALA1671823 | cell-based format | Scientific Literature | |
| 17. | ALA1679958 | F | Antagonist activity at human recombinant GABAb 1b/2 receptor expressed in Xenopus laevis oocytes co-expressing GIRK1/4 assessed as inhibition of GABA-induced current at 300 uM by two electrode voltage clamp technique | Homo sapiens | 1 | ALA1671823 | cell-based format | Scientific Literature | |
| 18. | ALA1679959 | F | Antagonist activity at human recombinant GABAb 1b/2 receptor expressed in Xenopus laevis oocytes co-expressing GIRK1/4 assessed as inhibition of GABA-induced current at 100 uM by two electrode voltage clamp technique | Homo sapiens | 2 | ALA1671823 | cell-based format | Scientific Literature | |
| 19. | ALA1679960 | F | Antagonist activity at human recombinant GABAb 1b/2 receptor expressed in Xenopus laevis oocytes co-expressing GIRK1/4 assessed as inhibition of GABA-induced current at 600 uM by two electrode voltage clamp technique | Homo sapiens | 2 | ALA1671823 | cell-based format | Scientific Literature | |
| 20. | ALA1680097 | F | Agonist activity at human recombinant GABAb 1b/2 receptor expressed in Xenopus laevis oocytes co-expressing GIRK1/4 assessed as inhibition of GABA-induced current by two electrode voltage clamp technique | Homo sapiens | 1 | ALA1671823 | cell-based format | Scientific Literature |
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