# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA653007 | B | Concentration required to displace 0.4 nM [3H]SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulfonyl fluoride | 7 | tissue-based format | Scientific Literature | |||
2. | ALA653008 | B | Concentration required to displace 0.4 nM [3H]SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulfonyl fluoride; Not tested | 2 | tissue-based format | Scientific Literature | |||
3. | ALA660010 | B | Binding affinity towards cannabinoid CB1 receptor in rat brain membrane by displacement of [3H]SR-141,716A | 12 | cell membrane format | Scientific Literature | |||
4. | ALA660011 | B | Binding affinity towards cannabinoid CB1 receptor in rat brain membrane by displacement of [3H]SR-141,716A at 50 uM | 2 | cell membrane format | Scientific Literature | |||
5. | ALA660012 | B | Binding affinity towards CB1 receptor in rat brain membrane by displacement of [3H]SR-141,716A relative to HU-210 | 14 | cell membrane format | Scientific Literature | |||
6. | ALA657996 | B | Inhibitory activity, measured by displacement [3H]CP-55940 from cannabinoid receptor (CB1) in rat brain | 44 | tissue-based format | Scientific Literature | |||
7. | ALA657997 | B | Binding affinity for the Cannabinoid receptor using [3H]CP-55940 as radioligand | 1 | single protein format | Scientific Literature | |||
8. | ALA661059 | B | Binding affinity for the cannabinoid brain receptor (CB1) using [3H]CP-55940 | 3 | assay format | Scientific Literature | |||
9. | ALA661060 | B | Compound was evaluated for binding affinity to displace [3H]CP-55940 radioligand from cannabinoid receptor in rat brain P2 membrane | 1 | cell membrane format | Scientific Literature | |||
10. | ALA661061 | B | Compound was evaluated for binding affinity towards cannabinoid receptor in rat brain P2 membrane | 1 | cell membrane format | Scientific Literature | |||
11. | ALA858284 | F | Cannabinoid receptor 1 dependent activity of compound was evaluated by using [35S]GTP-gamma-S-binding studies | 3 | assay format | Scientific Literature | |||
12. | ALA658202 | B | Percentage affinity towards Cannabinoid receptor 1 using [3H]CP-55940 as radioligand in rat forebrain membranes | 5 | cell membrane format | Scientific Literature | |||
13. | ALA658203 | F | Effective concentration for inhibition of Cannabinoid receptor 1-mediated adenylyl cyclase activity using African green monkey (COS-7) cells transfected with the cDNA of rat CB1 receptor | 12 | assay format | Scientific Literature | |||
14. | ALA884421 | F | In vivo effective dose to antagonise cannabinoid receptor 1 agonist (CP-55940) induced hypotension in rat upon peroral administration | 10 | organism-based format | Scientific Literature | |||
15. | ALA657117 | F | Maximal response of cannabinoid receptor to compound was evaluated using [35S]GTP-gamma-S-binding studies | 3 | assay format | Scientific Literature | |||
16. | ALA657118 | B | Binding affinity against brain Cannabinoid receptor 1 using [3H]CP-55940 as radioligand at 1.1 nM concentration | 2 | assay format | Scientific Literature | |||
17. | ALA657119 | B | Binding affinity against brain cannabinoid receptor 1 using [3H]CP-55940 as radioligand at 0.25 nM concentration | 5 | assay format | Scientific Literature | |||
18. | ALA657120 | B | Binding affinity towards Cannabinoid receptor 1 was determined using [3H]-CP- cannabinoid as radioligand with rat brain membrane | 3 | assay format | Scientific Literature | |||
19. | ALA657121 | B | Binding affinity towards Cannabinoid receptor 1 was determined using [3H]-CP- cannabinoid as radioligand with rat brain membrane in the presence of PMSF | 1 | assay format | Scientific Literature | |||
20. | ALA658880 | B | Concentration of compound required to inhibit 50% of [3H]WIN-55212 binding to Cannabinoid receptor 1 in rat cerebellum membranes. | 61 | cell membrane format | Scientific Literature |