| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA843623 | B | Selectivity for human PPAR delta over PPAR gamma receptor | Homo sapiens | 1 | protein format | Scientific Literature | ||
| 2. | ALA855871 | B | Selectivity for human PPARdelta over human PPARgamma | Homo sapiens | 2 | protein format | Scientific Literature | ||
| 3. | ALA855872 | B | Selectivity for human PPARdelta over human PPARgamma | Homo sapiens | 1 | protein format | Scientific Literature | ||
| 4. | ALA886019 | B | Selectivity for PPARdelta over PPARgamma | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 5. | ALA889307 | B | Selectivity for PPARgamma over PPARdelta | Homo sapiens | 20 | assay format | Scientific Literature | ||
| 6. | ALA1173894 | B | Activation of PPARbeta/gamma in human HaCaT cells assessed as induction of ANGPTL4 expression by PCR | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA1173895 | B | Activation of PPARbeta/gamma in human HaCaT cells assessed as inhibition of cellular proliferation at 10 uM after 72 hrs | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA1647907 | B | Selectivity ratio of EC50 for human PPARgamma DNA binding domain to EC50 for PPARdelta DNA binding domain | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 9. | ALA1648159 | B | Selectivity ratio of EC50 for full length human PPARgamma to EC50 for full length human PPARdelta | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA1936616 | B | Selectivity ratio of EC50 for human PPARdelta to EC50 for human PPARgamma1 | Homo sapiens | 11 | assay format | Scientific Literature | ||
| 11. | ALA2038125 | B | Selectivity ratio of EC50 for human PPARgamma to EC50 for human PPARdelta | Homo sapiens | 9 | assay format | Scientific Literature | ||
| 12. | ALA2067039 | B | Selectivity ratio of EC50 for PPARdelta LBD to EC50 for PPARgamma LBD | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 13. | ALA2162359 | B | Selectivity ratio of EC50 for human PPARdelta expressed in human HEK293 cells to EC50 for human PPARgamma expressed in human HEK293 cells | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 14. | ALA3395313 | B | Selectivity index, ratio of EC50 for Gal4-tagged PPARgamma ligand binding domain (unknown origin) to EC50 for Gal4-tagged PPARdelta ligand binding domain (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA3792247 | B | Ratio of EC50 for human PPAR gamma to EC50 for human PPAR delta | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 16. | ALA4184454 | B | Selectivity ratio of EC50 for GAL4-fused human PPARgamma LBD expressed in African green monkey CV1 cells to EC50 for GAL4-fused human PPARdelta LBD expressed in African green monkey CV1 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA4186886 | B | Selectivity ratio of IC50 for PPARdelta (unknown origin) to IC50 for RORgammat in human Jurkat cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA4307151 | B | Selectivity index, ratio of EC50 of PPARgamma (unknown origin) to EC50 of PPARdelta (unknown origin) | Homo sapiens | 3 | protein format | Scientific Literature | ||
| 19. | ALA4332112 | B | Selectivity ratio of IC50 for PPARdelta (unknown origin) to IC50 for PPARgamma (unknown origin) | Homo sapiens | 1 | protein format | Scientific Literature | ||
| 20. | ALA4359348 | B | Selectivity ratio of EC50 for partial agonist activity at Gal4-fused PPARdelta LBD (unknown origin) expressed in HEK293T cells to EC50 for partial agonist activity at Gal4-fused PPARgamma LBD (unknown origin) expressed in HEK293T cells | Homo sapiens | 1 | cell-based format | Scientific Literature |
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