| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA656373 | F | Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha; values in the parentheses indicates 95% confidence interval | 1 | ALA1135907 | cell-based format | Scientific Literature | ||
| 2. | ALA656374 | F | Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha | 5 | ALA1135907 | cell-based format | Scientific Literature | ||
| 3. | ALA651610 | F | Transcriptional activity against RXR:PPAR-gamma synergy was determined in vitro | Cercopithecidae | 17 | ALA1145809 | assay format | Scientific Literature | |
| 4. | ALA658488 | F | Synergistic efficacy against RXR:PPAR-gamma heterodimer was determined in vitro | Cercopithecidae | 17 | ALA1145809 | assay format | Scientific Literature | |
| 5. | ALA659132 | F | Synergistic efficacy for RXR and PPAR-gamma heterodimer in vitro; Not applicable | Cercopithecidae | 1 | ALA1145809 | assay format | Scientific Literature | |
| 6. | ALA659133 | F | Synergistic transcriptional activation of RXR and PPAR-gamma heterodimer in vitro; Not applicable | Cercopithecidae | 1 | ALA1145809 | assay format | Scientific Literature | |
| 7. | ALA759726 | F | Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha | Homo sapiens | 1 | ALA1135907 | cell-based format | Scientific Literature | |
| 8. | ALA772126 | F | Synergistic activation of BRL-49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assay | Homo sapiens | 9 | ALA1136229 | cell-based format | Scientific Literature | |
| 9. | ALA772127 | F | Synergistic activation of BRL-49653 mediated PPAR gamma and retinoid X receptor alpha expressed in CV-1 cell transcriptional activation assay | Homo sapiens | 9 | ALA1136229 | cell-based format | Scientific Literature | |
| 10. | ALA1227770 | B | Transactivation of PPARgamma/RXRalpha heterodimer | 3 | ALA1221250 | protein complex format | Scientific Literature | ||
| 11. | ALA1696526 | F | Agonist activity at PPARgamma/RXRalpha transfected in human COS1 cells at 10'-7 to 10'-6 M after 18 hrs by luciferase reporter gene transactivation assay | 2 | ALA1687703 | cell-based format | Scientific Literature | ||
| 12. | ALA2149517 | F | Agonist activity at PPARgamma/RXRalpha expressed in human Cos1 cells after 18 hrs by SEAP reporter gene assay | Homo sapiens | 3 | ALA2146420 | cell-based format | Scientific Literature | |
| 13. | ALA2341868 | B | Transactivation of PPARgamma/RXRalpha (unknown origin) by luciferase reporter gene assay relative to TIPP703 | Homo sapiens | 1 | ALA2331224 | protein complex format | Scientific Literature | |
| 14. | ALA4340395 | B | Induction of RXRalpha/PPARgamma interaction in HUVEC at 10 uM pretreated for 20 hrs before TNFalpha stimulation by immunoprecipitation and Western blotting analysis | Homo sapiens | 1 | ALA4339250 | cell-based format | Scientific Literature | |
| 15. | ALA4340396 | B | Induction of RXRalpha/PPARgamma interaction in HUVEC at 1 uM pretreated for 20 hrs before TNFalpha stimulation by immunoprecipitation and Western blotting analysis | Homo sapiens | 1 | ALA4339250 | cell-based format | Scientific Literature | |
| 16. | ALA4359358 | B | Partial agonist activity at 1:1 Gal4-fused PPARgamma LBD/Gal4-fused RXRalpha (unknown origin) expressed in HEK293T cells after 14 to 16 hrs by dual-Glo luciferase assay | Homo sapiens | 1 | ALA4354876 | cell-based format | Scientific Literature | |
| 17. | ALA4359359 | B | Partial agonist activity at 1:2 Gal4-fused PPARgamma LBD/Gal4-fused RXRalpha (unknown origin) expressed in HEK293T cells at 0.1 to 1 uM after 14 to 16 hrs by dual-Glo luciferase assay | Homo sapiens | 1 | ALA4354876 | cell-based format | Scientific Literature | |
| 18. | ALA4414350 | B | Activation of full-length RXRalpha/PPARgamma (unknown origin) transfected in HEK293T cells at 30 uM after 12 to 14 hrs by dual-glo luciferase reporter gene assay | Homo sapiens | 1 | ALA4411340 | cell-based format | Scientific Literature | |
| 19. | ALA4414351 | B | Activation of PPARgamma/RXRalpha in human HepG2 cells assessed as increase in ANGPTL4 mRNA expression at 30 uM after 12 hrs followed by renewal of medium containing test compounds after 6 hrs by PCR analysis | Homo sapiens | 1 | ALA4411340 | cell-based format | Scientific Literature | |
| 20. | ALA4414352 | B | Activation of PPARgamma/RXRalpha in human HepG2 cells assessed as increase in ANGPTL4 mRNA expression at 10 uM after 12 hrs followed by renewal of medium containing test compounds after 6 hrs by PCR analysis | Homo sapiens | 1 | ALA4411340 | cell-based format | Scientific Literature |
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