| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA929248 | B | Displacement of fluorescent 5-(3-(3-(4-((4-((7-(hydroxyamino)-7-oxoheptyl)carbamoyl)phenylamino)methyl)-1H-1,2,3-triazol-1-yl)propyl)thioureido)-2-(3-hydroxy-6-oxo-6H-xanthen-9-yl)benzoic acid from human HDAC3/NcoR2 by fluorescence polarization assay | Homo sapiens | 7 | ALA1145631 | protein complex format | Scientific Literature | |
| 2. | ALA1772081 | B | Inhibition of full length HDAC3/NCoR2 assessed as 7-amino-4-methylcoumarin release from fluorophore conjugated substrate after 5 mins by fluorescence assay | 6 | ALA1770095 | protein complex format | Scientific Literature | ||
| 3. | ALA1838189 | B | Inhibition of recombinant human HDAC3/NCOR2 using Boc-L-Lys(epsilon-trifluoroacetyl)-AMC as substrate by two-step fluorogenic assay | Homo sapiens | 6 | ALA1833850 | protein complex format | Scientific Literature | |
| 4. | ALA1838195 | B | Inhibition of recombinant human HDAC3/N-CoR2 using Boc-L-Lys(epsilon-trifluoroacetyl)-AMC as substrate by two-step fluorogenic assay in presence of 0.2 mM H2O2 (Rvb = 0.018 uM) | Homo sapiens | 1 | ALA1833850 | protein complex format | Scientific Literature | |
| 5. | ALA1838196 | B | Inhibition of recombinant human HDAC3/N-CoR2 using Boc-L-Lys(epsilon-trifluoroacetyl)-AMC as substrate by two-step fluorogenic assay in presence of 0.4 mM H2O2 (Rvb = 0.018 uM) | Homo sapiens | 1 | ALA1833850 | protein complex format | Scientific Literature | |
| 6. | ALA1838197 | B | Inhibition of recombinant human HDAC3/N-CoR2 using Boc-L-Lys(epsilon-trifluoroacetyl)-AMC as substrate by two-step fluorogenic assay in presence of 1 mM H2O2 (Rvb = 0.018 uM) | Homo sapiens | 1 | ALA1833850 | protein complex format | Scientific Literature | |
| 7. | ALA1920770 | B | Selectivity ratio of compound IC50 to SAHA IC50 for human recombinant HDAC3/NCoR2 using fluorophore-conjugated substrate Boc-L-Lys(Ac)-AMC after 60 mins | Homo sapiens | 2 | ALA1914352 | protein complex format | Scientific Literature | |
| 8. | ALA1921157 | B | Inhibition of human recombinant HDAC3/NCoR2 using fluorophore-conjugated substrate Boc-L-Lys(Ac)-AMC | Homo sapiens | 10 | ALA1914352 | protein complex format | Scientific Literature | |
| 9. | ALA2014703 | B | Inhibition of recombinant human HDAC3-NCoR2 using Fluor-de-Lys as substrate after 30 mins by spectrophotometry | Homo sapiens | 2 | ALA2010669 | protein complex format | Scientific Literature | |
| 10. | ALA2014771 | B | Inhibition of HDAC3-NCoR2 in human HeLa cells nuclear extract using Fluor-de-Lys as substrate after 30 mins by spectrophotometry | Homo sapiens | 18 | ALA2010669 | cell-based format | Scientific Literature | |
| 11. | ALA2065939 | B | Inhibition of recombinant HDAC3/NCoR2 at 1 uM | Homo sapiens | 1 | ALA2062402 | protein complex format | Scientific Literature | |
| 12. | ALA2065942 | B | Inhibition of recombinant HDAC3/NCoR2 using Ac-Lys(Ac)-AMC as substrate after 30 mins by fluorescence analysis | Homo sapiens | 4 | ALA2062402 | protein complex format | Scientific Literature | |
| 13. | ALA2065946 | B | Ratio of IC50 for valproic acid to compound for recombinant HDAC3/NCoR2 using Ac-Lys(Ac)-AMC as substrate after 30 mins by fluorescence analysis | Homo sapiens | 1 | ALA2062402 | protein complex format | Scientific Literature | |
| 14. | ALA2065957 | B | Competitive inhibition of HDAC3/NCoR2 using Ac-Lys(Ac)-AMC as substrate by Lineweaver-Burk plot analysis | Homo sapiens | 1 | ALA2062402 | protein complex format | Scientific Literature | |
| 15. | ALA2065959 | B | Inhibition of recombinant HDAC3/NCoR2 at 10 uM | Homo sapiens | 1 | ALA2062402 | protein complex format | Scientific Literature | |
| 16. | ALA2174034 | B | Inhibition of human recombinant HDAC3/NCoR2 using Ac-Lys(Ac)-7-amino-4-methylcoumarin as substrate after 30 mins by trypsin-coupled fluorogenic assay | Homo sapiens | 6 | ALA2169795 | protein complex format | Scientific Literature | |
| 17. | ALA2399517 | B | Inhibition of HDAC3/NCOR2 (unknown origin) using Arg-His-Lys-Lys(Ac) as substrate assessed as residual activity at 3.3 x 10'-5 M after 2 hrs by fluorescence assay relative to control | Homo sapiens | 4 | ALA2396570 | protein complex format | Scientific Literature | |
| 18. | ALA2424317 | B | Inhibition of HDAC3/NcoR2 (unknown origin) using RHKKAc from p53 as substrate | Homo sapiens | 2 | ALA2417402 | protein complex format | Scientific Literature | |
| 19. | ALA2432125 | B | Inhibition of HDAC3/NcoR2 (unknown origin) using RHKKAc as substrate | Homo sapiens | 2 | ALA2429834 | protein complex format | Scientific Literature | |
| 20. | ALA3102464 | B | Inhibition of human HDAC3/NCOR2 using RHKK(Ac) as substrate by fluorimetric analysis | Homo sapiens | 19 | ALA3098008 | protein complex format | Scientific Literature |
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