#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA3537619	ADME	Activation of PXR in rat hepatocytes assessed as increase in CYP3A-mediated testosterone 6beta-hydroxylation at 10 uM after 24 hrs by HPLC analysis relative to control	Rattus norvegicus	1	ALA3526076	cell-based format	Scientific Literature
2.	ALA3532960	ADME	Antagonist activity at rat PXR expressed in human HepG2 cells coexpressing CYP3A4 assessed as inhibition of PCN-induced receptor activation up to 100 uM after 24 hrs by dual luciferase reporter gene assay	Rattus norvegicus	1	ALA3526076	cell-based format	Scientific Literature
3.	ALA3532963	ADME	Antagonist activity at rat PXR expressed in human HepG2 cells coexpressing CYP3A4 assessed as inhibition of PCN-induced receptor activation at 30 uM after 24 hrs by dual luciferase reporter gene assay	Rattus norvegicus	1	ALA3526076	cell-based format	Scientific Literature
4.	ALA3531874	ADME	Activation of rat PXR expressed in human HepG2 cells after 24 hrs by luciferase reporter gene based luminescent analysis	Rattus norvegicus	36	ALA3525965	cell-based format	Scientific Literature
5.	ALA3531877	ADME	Activation of rat PXR expressed in human HepG2 cells up to 46 uM after 24 hrs by luciferase reporter gene based luminescent analysis	Rattus norvegicus	41	ALA3525965	cell-based format	Scientific Literature
6.	ALA3531881	ADME	Activation of rat PXR expressed in human HepG2 cells after 24 hrs by luciferase reporter gene based luminescent analysis relative to dexamethasone	Rattus norvegicus	31	ALA3525965	cell-based format	Scientific Literature
7.	ALA3532296	ADME	Activation of rat PXR expressed in rat hepatocytes coexpressing CYP3A4 at 100 uM after 24 hrs by dual luciferase reporter gene assay	Rattus norvegicus	1	ALA3526076	cell-based format	Scientific Literature
8.	ALA3532297	ADME	Activation of rat PXR expressed in rat hepatocytes coexpressing CYP3A4 at 10 uM after 24 hrs by dual luciferase reporter gene assay relative to control	Rattus norvegicus	2	ALA3526076	cell-based format	Scientific Literature
9.	ALA3532298	ADME	Activation of rat PXR expressed in human HepG2 cells coexpressing CYP3A4 at 0.1 to 100 uM after 24 hrs by dual luciferase reporter gene assay	Rattus norvegicus	1	ALA3526076	cell-based format	Scientific Literature
10.	ALA3532299	ADME	Activation of rat PXR expressed in human HepG2 cells coexpressing CYP3A4 at 0.1 to 10 uM after 24 hrs by dual luciferase reporter gene assay relative to control	Rattus norvegicus	2	ALA3526076	cell-based format	Scientific Literature
11.	ALA3532304	ADME	Activation of PXR in rat hepatocytes assessed as upregulation of CYP3A23 mRNA expression at 1 to 30 uM after 24 hrs by RT-PCR analysis	Rattus norvegicus	1	ALA3526076	cell-based format	Scientific Literature
12.	ALA3532305	ADME	Activation of PXR in rat hepatocytes assessed as upregulation of CYP3A23 mRNA expression at 10 uM after 24 hrs by RT-PCR analysis relative to control	Rattus norvegicus	1	ALA3526076	cell-based format	Scientific Literature
13.	ALA3532306	ADME	Activation of PXR in rat hepatocytes assessed as effect on CYP3A-mediated testosterone 6beta-hydroxylation at 1 to 30 uM after 24 hrs by HPLC analysis	Rattus norvegicus	1	ALA3526076	cell-based format	Scientific Literature
14.	ALA3528709	ADME	Transactivation of rat PXR at 0.1 to 30 uM after 24 to 48 hrs by cell-based luciferase reporter gene assay	Rattus norvegicus	3	ALA3526135	cell-based format	Scientific Literature
15.	ALA1217433	Binding	Activation of rat PXR	Rattus norvegicus	1	ALA1212831	single protein format	Scientific Literature
16.	ALA2114797	Functional	PubChem BioAssay. qHTS assay for small molecule activators of the rat pregnane X receptor (rPXR) signaling pathway. (Class of assay: confirmatory)	Rattus norvegicus	424	ALA1201862	assay format	PubChem BioAssays
17.	ALA2384332	Binding	Activation of rat PXR at 10 uM relative to control	Rattus norvegicus	3	ALA2380263	single protein format	Scientific Literature
18.	ALA5051538	Binding	Activation of rat pregnane X receptor at 10 uM relative to control	Rattus norvegicus	1	ALA5050846	single protein format	Patent Bioactivity Data
19.	ALA5105656	Binding	Activation of rat PXR assessed as induction of PXR activity at 10 uM relative to control	Rattus norvegicus	17	ALA5104129	single protein format	Scientific Literature
20.	ALA5258194	Binding	Activation of rat PXR	Rattus norvegicus	1	ALA5257040	single protein format	Scientific Literature