| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2156127 | F | Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level by FLIPR assay | Homo sapiens | 47 | cell-based format | Scientific Literature | ||
| 2. | ALA2155422 | F | Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at 10 uM by FLIPR assay | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 3. | ALA4729958 | F | Antagonist activity at human SUCNR1 expressed in human CHEM1 cells incubated for 60 mins in presence of [35S]GTPgammaS by scintillation proximity assay | Homo sapiens | 19 | cell-based format | Scientific Literature | ||
| 4. | ALA4729960 | F | Antagonist activity at human SUCNR1 expressed in human CHEM1 cell membranes at 100 uM incubated for 60 mins in presence of [35S]GTPgammaS by scintillation proximity assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA4883603 | B | PRESTO-Tango GPCRome screening (SUCNR1) | 1 | single protein format | Donated Chemical Probes - SGC Frankfurt |
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