# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2167521 | B | Inhibition of human KDM7A catalytic domain expressed in Escherichia coli by MALDI assay | Homo sapiens | 1 | ALA2163321 | assay format | Scientific Literature | |
2. | ALA2427597 | B | Inhibition of KDM7A in human HeLa cells assessed as down-regulation of E2F1 mRNA expressing at 80 uM by RT-PCR analysis | Homo sapiens | 1 | ALA2424657 | cell-based format | Scientific Literature | |
3. | ALA2427604 | B | Inhibition of KDM7A (unknown origin) using K27me2 peptide as substrate by MALDI assay | Homo sapiens | 4 | ALA2424657 | single protein format | Scientific Literature | |
4. | ALA4122975 | B | Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by peptide addition measured after 1 hr by luminescence-based AlphaScreen assay | Homo sapiens | 15 | ALA4118181 | single protein format | Scientific Literature | |
5. | ALA4122979 | B | Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed by peptide addition measured after 1 hr by luminescence-based AlphaScreen assay | Homo sapiens | 6 | ALA4118181 | single protein format | Scientific Literature | |
6. | ALA4122980 | B | Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) at 100 uM preincubated for 15 mins followed by peptide addition measured after 1 hr by luminescence-based AlphaScreen assay | Homo sapiens | 1 | ALA4118181 | single protein format | Scientific Literature | |
7. | ALA4122981 | B | Inhibition of KDM7A (PHD-JmjC) (unknown origin) demethylation activity at 100 uM preincubated for 10 mins followed by H3(1-15)K9me2 peptide substrate addition by MALDI-TOF-MS analysis | Homo sapiens | 7 | ALA4118181 | single protein format | Scientific Literature |