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# Aladdin ID Assay Type Description Organism Compounds Reference BAO Format Source 1. ALA666530 F Effective concentration to inhibit D216,ND217N,E218Q KL-2 Opioid receptor kappa 1 binding to [35S]GTP-gamma-S, expressed in COS cells 1 cell-based format Scientific Literature 2. ALA666531 B Dissociation constant against D216N,D217N,E218Q EL-2 Opioid receptor kappa 1 expressed in HEK cells 1 cell-based format Scientific Literature 3. ALA663515 B Binding constant against D216N,D217N,E218Q EL-2 Opioid receptor kappa 1 using [3H]diprenorphine as radioligand expressed in HEK cells 2 cell-based format Scientific Literature 4. ALA679838 B Dissociation constant against E203Q,D204N,D206N EL-2 Opioid receptor kappa 1 expressed in HEK cells 1 cell-based format Scientific Literature 5. ALA679839 B Binding constant against E203Q,D204N,D206N EL-2 Opioid receptor kappa 1 using [3H]diprenorphine as radioligand expressed in HEK cells 2 cell-based format Scientific Literature 6. ALA679840 F Effective concentration to inhibit E203Q,D204N,D206N KL-2 Opioid receptor kappa 1 binding to [35S]GTP-gamma-S, expressed in COS cells 1 cell-based format Scientific Literature 7. ALA679841 B Dissociation constant against E203Q,D204N,D206N,E209Q EL-2 Opioid receptor kappa 1 expressed in HEK cells 1 cell-based format Scientific Literature 8. ALA679842 B Binding constant against E203Q,D204N,D206N,E209Q EL-2 Opioid receptor kappa 1 using [3H]diprenorphine as radioligand expressed in HEK cells 2 cell-based format Scientific Literature 9. ALA677621 F Effective concentration to inhibit E203Q,D204N,D206N,E209Q KL-2 Opioid receptor kappa 1 binding to [35S]GTP-gamma-S, expressed in COS cells 1 cell-based format Scientific Literature 10. ALA700237 B Binding affinity against rat kappa-opioid receptor expressed in CHO cells was determined by competitive inhibition of 2 nM [3H]-U 69593 Rattus norvegicus 9 cell-based format Scientific Literature 11. ALA753141 B Binding ability towards opioid receptor kappa expressed in homogenates of rat brain. 9 tissue-based format Scientific Literature 12. ALA753142 B The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]DADLE 4 single protein format Scientific Literature 13. ALA753143 B The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]naloxone 4 single protein format Scientific Literature 14. ALA753144 B Ratio of IC50 of opioid receptor kappa to IC50 opioid receptor mu 9 single protein format Scientific Literature 15. ALA753315 F Effective concentration to inhibit wild type KL-2 Opioid receptor kappa 1 binding to [35S]GTP-gamma-S, expressed in COS cells 1 cell-based format Scientific Literature 16. ALA753316 F Inhibition of Forskolin-Stimulated Adenylyl Cyclase in CHO cells expressing Opioid receptor kappa 1 Rattus norvegicus 9 cell-based format Scientific Literature 17. ALA753317 F Inhibition of forskolin-stimulated adenylyl cyclase activity by compound in CHO cells expressing Opioid receptor kappa 1 6 cell-based format Scientific Literature 18. ALA753318 B Effect on binding affinity of mutational exchange of Glu297 in the Opioid receptor kappa 1 in transiently expressed rat cos-7 cells activity expressed as binding ratio with nor-BNI. 3 assay format Scientific Literature 19. ALA753319 B Mutant factor against mutant receptor with Opioid receptor kappa 1 3 single protein format Scientific Literature 20. ALA753902 B Inhibitory concentration was evaluated against kappa opioid receptor by displacement of tritiated U-69593 from rat brain membranes 8 cell membrane format Scientific Literature