# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2186997 | B | Inhibition of His6FLAG-tagged TRIM33 isoform B expressed in Escherichia coli assessed as change in melting temperature at 100 uM by thermal shift assay | 2 | ALA2176978 | assay format | Scientific Literature | ||
2. | ALA3383434 | B | Inhibition of human TIF1gamma PHD/bromodomain by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
3. | ALA3383435 | B | Inhibition of human WDR2 bromodomain 2 by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
4. | ALA3825927 | B | Binding affinity to His6-tagged human recombinant TRIM33B bromodomain expressed in Escherichia coli BL21(DE3)-R3-pRARE2 cells assessed as change in melting temperature at 10 uM by SyproOrange dye based DSF thermal shift assay | Homo sapiens | 1 | ALA3822370 | cell-based format | Scientific Literature | |
5. | ALA4020278 | B | Binding affinity to human TRIM33 (PHD, Bromo) (D882 to A1087 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 1 | ALA4017535 | assay format | Scientific Literature | |
6. | ALA4038420 | B | Inhibition of human TRIM33-phd-bromo (D882 to A1087 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 3 | ALA4038268 | assay format | Scientific Literature | |
7. | ALA4047559 | B | Inhibition of human partial length TRIM33-phd-bromo (D882 to A1087 residues) expressed in bacterial expression system assessed as residual activity at 500 nM relative to control by BROMOscan assay | Homo sapiens | 1 | ALA4043246 | assay format | Scientific Literature | |
8. | ALA4053071 | B | Inhibition of human TRIM33 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assay | Homo sapiens | 1 | ALA4052588 | assay format | Scientific Literature | |
9. | ALA4118630 | B | Binding affinity to TRIM33 in human NCI-H23 cells at 1 uM by mass spectrometry based pull down assay | Homo sapiens | 1 | ALA4118021 | cell-based format | Scientific Literature | |
10. | ALA4130878 | B | Inhibition of human partial length TRIM33 (D882 to A1087 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1 uM after 1 hr by qPCR method relative to control | Homo sapiens | 1 | ALA4130345 | assay format | Scientific Literature | |
11. | ALA4151046 | B | Binding affinity to human TRIM33-phd-bromo (D882 to A1087 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 1 | ALA4145654 | assay format | Scientific Literature | |
12. | ALA4186442 | B | Binding affinity to human partial length TRIM33 (D882 to A1087 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 1 | ALA4184171 | assay format | Scientific Literature | |
13. | ALA4189334 | B | Binding affinity to human partial length DNA-tagged TRIM33(PHD,Bromo.) expressed in bacteria by BROMOscan method | Homo sapiens | 1 | ALA4184317 | assay format | Scientific Literature | |
14. | ALA4194927 | B | Binding affinity to human TRIM33-phd-bromo expressed in bacterial system assessed as remaining binding level at 1 uM by BROMOscan assay relative to control | Homo sapiens | 3 | ALA4190379 | assay format | Scientific Literature | |
15. | ALA4198534 | B | Inhibition of human TRIM33-phd-bromodomain (D882 to A1087 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1 uM after 1 hr by BROMOScan assay relative to control | Homo sapiens | 1 | ALA4196075 | assay format | Scientific Literature | |
16. | ALA4332550 | B | Binding affinity to human partial length TRIM33 PHD bromodomain (D882 to A1087 residues) expressed in bacterial expression system after 1 hr by bromoscan assay | Homo sapiens | 1 | ALA4330118 | assay format | Scientific Literature | |
17. | ALA4351664 | B | Binding affinity to human partial length TRIM33 (D882 to A1087 residues) expressed in bacterial expression system at 1 uM by BROMOscan assay | Homo sapiens | 1 | ALA4350961 | assay format | Scientific Literature | |
18. | ALA4415511 | B | Binding affinity to human partial length TRIM33 (D882 to A1087 residues) expressed in Escherichia coli BL21 cells assessed as residual binding level at 1 uM measured after 1 hr by quantitative PCR based BROMOscan assay relative to control | Homo sapiens | 1 | ALA4414574 | cell-based format | Scientific Literature | |
19. | ALA4418855 | B | Inhibition of recombinant TRIM33 PHD bromodomain (unknown origin) using biotinylated H3 peptide (H3K9me3K18ac) by AlphaScreen assay | Homo sapiens | 110 | ALA4418499 | single protein format | Patent Bioactivity Data | |
20. | ALA4612517 | B | Binding affinity to human partial length TRIM33 phd bromodomain (D882 to A1087 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 1 | ALA4610112 | assay format | Scientific Literature |