# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2186999 | B | Inhibition of His6FLAG-tagged BRD1 expressed in Escherichia coli assessed as change in melting temperature at 100 uM by thermal shift assay | 2 | ALA2176978 | assay format | Scientific Literature | ||
2. | ALA3267586 | B | Binding affinity to BRD1 (unknown origin) by thermal shift assay | Homo sapiens | 2 | ALA3259646 | single protein format | Scientific Literature | |
3. | ALA3385106 | B | Binding affinity to 6H-Flag-tagged Tev-BRPF2 (551-673 aa) (unknown origin) by TR-FRET competitive assay | Homo sapiens | 1 | ALA3352488 | single protein format | Scientific Literature | |
4. | ALA3383437 | B | Inhibition of human BRD1 by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
5. | ALA3591380 | B | Binding affinity to BRPF2 (unknown origin) by BROMOscan panel based assay | Homo sapiens | 1 | ALA3588744 | single protein format | Scientific Literature | |
6. | ALA3743451 | B | Binding affinity to human BRD1 at 10 uM by differential scanning fluorimetry | Homo sapiens | 1 | ALA3739345 | single protein format | Scientific Literature | |
7. | ALA3757234 | B | Binding affinity to BRPF2 (unknown origin) by isothermal titration calorimetry | Homo sapiens | 1 | ALA3751772 | single protein format | Scientific Literature | |
8. | ALA3773110 | B | Binding affinity to biotinylated BRD1 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
9. | ALA3771490 | B | Inhibition of BRPF2 BRD1 (unknown origin) by Alpha Screen assay | Homo sapiens | 25 | ALA3769336 | single protein format | Scientific Literature | |
10. | ALA3771493 | B | Binding affinity to BRPF2 BRD1 (unknown origin) by isothermal titration calorimetry | Homo sapiens | 1 | ALA3769336 | single protein format | Scientific Literature | |
11. | ALA3779322 | B | Binding affinity to recombinant human BRPF2 expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
12. | ALA3782669 | B | Binding affinity to human His6-tagged BRD1 (E556 to A688 residues) expressed in Escherichia coli BL21(DE3) cells at 200 uM incubated for 30 mins by SYPRO orange staining based fluorescence thermal shift assay | Homo sapiens | 16 | ALA3779865 | cell-based format | Scientific Literature | |
13. | ALA3790874 | B | Binding affinity to BRPF2 (unknown origin) by isothermal titration calorimetric analysis | Homo sapiens | 2 | ALA3785033 | single protein format | Scientific Literature | |
14. | ALA3830585 | B | Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6HisFlag-Tev-BRPF2 (551 to 673 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells after 30 mins by TR-FRET assay | Homo sapiens | 2 | ALA3826893 | cell-based format | Scientific Literature | |
15. | ALA3863024 | B | Binding affinity to BRD1 (unknown origin) assessed as change in melting temperature at 100 uM by differential scanning fluorimetric assay | Homo sapiens | 1 | ALA3861991 | single protein format | Scientific Literature | |
16. | ALA4030908 | B | Inhibition of human BRPF2 (556 to 688 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assay | Homo sapiens | 21 | ALA4028852 | assay format | Scientific Literature | |
17. | ALA4030916 | B | Inhibition of His-tagged BRPF2 (unknown origin) after 30 mins by alphaScreen assay | Homo sapiens | 1 | ALA4028852 | single protein format | Scientific Literature | |
18. | ALA4030940 | B | Binding affinity to BRPF2 (unknown origin) by isothermal titration calorimetry | Homo sapiens | 1 | ALA4028852 | single protein format | Scientific Literature | |
19. | ALA4030944 | B | Inhibition of GFP-BRD1 fusion construct (unknown origin) binding to chromatin by FRAP assay | Homo sapiens | 1 | ALA4028852 | single protein format | Scientific Literature | |
20. | ALA4038412 | B | Inhibition of human BRD1 (E556 to A688 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 2 | ALA4038268 | assay format | Scientific Literature |