| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA759509 | F | Antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 ) | 11 | ALA1135773 | assay format | Scientific Literature | ||
| 2. | ALA759510 | B | Affinity at P2X purinoceptor 1 (P2X1) and the value is expressed as IC50 | 1 | ALA1135726 | single protein format | Scientific Literature | ||
| 3. | ALA759511 | F | The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 1 (P2X1 ) | 1 | ALA1135773 | assay format | Scientific Literature | ||
| 4. | ALA874555 | F | Inhibitory concentration against human P2X purinoceptor 1 (hP2X1) expressed in CHO-K1 cells | Homo sapiens | 1 | ALA1139575 | cell-based format | Scientific Literature | |
| 5. | ALA872176 | F | Inhibitory concentration against human P2X purinoceptor 1 expressed in Xenopus laevis oocytes | Homo sapiens | 1 | ALA1140384 | cell-based format | Scientific Literature | |
| 6. | ALA901767 | B | Activity at human P2X1 receptor at 10 uM | Homo sapiens | 1 | ALA1138274 | single protein format | Scientific Literature | |
| 7. | ALA886465 | B | Activity at human P2X1 receptor at 10 uM | Homo sapiens | 1 | ALA1139969 | single protein format | Scientific Literature | |
| 8. | ALA1017977 | F | Antagonist activity at P2X1 receptor up to 10 uM | 1 | ALA1153300 | assay format | Scientific Literature | ||
| 9. | ALA960838 | B | Inhibition of P2X1 receptor | 1 | ALA1153301 | single protein format | Scientific Literature | ||
| 10. | ALA1069594 | F | Antagonist activity at P2X1 receptor | 2 | ALA1159093 | assay format | Scientific Literature | ||
| 11. | ALA2184468 | F | Antagonist activity at human P2X1 receptor by cell-based calcium influx assay | Homo sapiens | 8 | ALA2177033 | cell-based format | Scientific Literature | |
| 12. | ALA2184484 | F | Antagonist activity at human P2X1 receptor at 10 uM by cell-based calcium influx assay | Homo sapiens | 4 | ALA2177033 | cell-based format | Scientific Literature | |
| 13. | ALA2379686 | B | Antagonist activity at P2X1 receptor (unknown origin) | Homo sapiens | 1 | ALA2375299 | single protein format | Scientific Literature | |
| 14. | ALA3108480 | B | Antagonist activity at human P2X1 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP addition by Fluo-4 AM dye-based fluorescence assay | Homo sapiens | 6 | ALA3102848 | cell-based format | Scientific Literature | |
| 15. | ALA3107657 | B | Antagonist activity at P2X1 receptor in HEK293 cells assessed as alpha, beta-methylene ATP-induced calcium flux by FLIPR assay | Homo sapiens | 1 | ALA3102727 | cell-based format | Scientific Literature | |
| 16. | ALA3292927 | B | Antagonist activity at P2X1 receptor (unknown origin) by FLIPR assay | Homo sapiens | 1 | ALA3286275 | single protein format | Scientific Literature | |
| 17. | ALA3369083 | B | Antagonist activity against P2X1 (unknown origin) | Homo sapiens | 1 | ALA3351863 | single protein format | Scientific Literature | |
| 18. | ALA3744573 | B | Inhibition of P2X1R (unknown origin) | Homo sapiens | 1 | ALA3739255 | single protein format | Scientific Literature | |
| 19. | ALA3748119 | B | Agonist activity at human platelet P2X1 receptor assessed as increase in cytosolic calcium level at 1 uM by FLURO-4 staining based flow cytometric analysis relative to beta,gamma-CH2-ATP | Homo sapiens | 18 | ALA3745686 | assay format | Scientific Literature | |
| 20. | ALA4033446 | B | Activity at P2X1 (unknown origin) upto 10 uM by FLIPR assay | Homo sapiens | 2 | ALA4028916 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!