| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA751803 | F | The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 2 (P2X2) at 30 uM | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 2. | ALA751804 | F | The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 2 (P2X2) at 30 uM | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 3. | ALA751805 | F | The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 2 (P2X2) receptor 10 uM | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 4. | ALA759522 | F | The compound was evaluated for antagonist activity against recombinant human receptor P2X purinoceptor 2 (P2X2 ) | 3 | assay format | Scientific Literature | |||
| 5. | ALA759523 | F | The compound was evaluated for antagonist activity against recombinant human receptor P2X purinoceptor 2 (P2X2) | 1 | assay format | Scientific Literature | |||
| 6. | ALA759524 | B | KB value was evaluated at the human P2X purinoceptor 2 (P2X2); IA menas inactive | 1 | single protein format | Scientific Literature | |||
| 7. | ALA827768 | F | Inhibitory concentration against human P2X purinoceptor 2 (hP2X2) expressed in 1321N1 astrocytoma cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 8. | ALA931270 | B | Inhibition of P2X2 receptor | 1 | single protein format | Scientific Literature | |||
| 9. | ALA935655 | B | Displacement of [3H]alpha,beta-methyl ATP from P2X receptor | 1 | single protein format | Scientific Literature | |||
| 10. | ALA886466 | F | Antagonist activity at human P2X2 receptor at 10 uM | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA1017978 | F | Antagonist activity at P2X2 receptor up to 10 uM | 1 | assay format | Scientific Literature | |||
| 12. | ALA960839 | B | Inhibition of P2X2 receptor | 1 | single protein format | Scientific Literature | |||
| 13. | ALA1069595 | F | Antagonist activity at P2X2 receptor | 2 | assay format | Scientific Literature | |||
| 14. | ALA2184467 | F | Antagonist activity at human P2X2 receptor by cell-based calcium influx assay | Homo sapiens | 8 | cell-based format | Scientific Literature | ||
| 15. | ALA2184483 | F | Antagonist activity at human P2X2 receptor at 10 uM by cell-based calcium influx assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 16. | ALA2400256 | B | Activity at human recombinant purinergic P2X2 receptor expressed in Xenopus oocytes assessed as effect on ATP-induced activation at 3 uM by two-electrode voltage clamp technique relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA2427310 | B | Inhibition of human purinergic receptor P2X subunit-2 expressed in Xenopus laevis oocytes assessed as inhibition of ATP-induced current at 3 uM by two-electrode voltage clamp method | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 18. | ALA3108478 | B | Antagonist activity at human P2X2 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx at 100 uM preincubated for 30 mins followed by ATP addition by Fluo-4 AM dye-based fluorescence assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 19. | ALA3108479 | B | Antagonist activity at human P2X2 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubated for 30 mins followed by ATP addition by Fluo-4 AM dye-based fluorescence assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 20. | ALA3369084 | B | Antagonist activity against P2X2 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature |
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