| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA754458 | F | The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 7 (P2X7) | 2 | assay format | Scientific Literature | |||
| 2. | ALA754459 | F | The compound was evaluated for antagonist activity against P2X purinoceptor 7 (P2X7) in rat parotid acinar cells | 1 | cell-based format | Scientific Literature | |||
| 3. | ALA872175 | F | Inhibitory concentration against rat P2X purinoceptor 7 expressed in Xenopus laevis oocytes | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA869037 | F | Antagonist activity at rat P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of calcium flux by FLIPR | Rattus norvegicus | 10 | cell-based format | Scientific Literature | ||
| 5. | ALA1815873 | B | Inhibition of rat P2X7 by fluorescent-based live-cell assay | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 6. | ALA900721 | F | Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzoyl-ATP-induced changes in plasma membrane pore formation | Rattus norvegicus | 20 | cell-based format | Scientific Literature | ||
| 7. | ALA886456 | F | Antagonist activity at rat recombinant P2X7 receptor | Rattus norvegicus | 5 | assay format | Scientific Literature | ||
| 8. | ALA1680813 | F | Antagonist activity against rat P2X7 receptor expressed in Xenopus laevis oocyte assessed as inhibition of alpha, beta-meATP-induced inward current by two-electrode voltage-clamp electrophysiology | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 9. | ALA1804946 | F | Antagonist activity at rat recombinant P2X7 receptor expressed in HEK293 cells by ethidium bromide release assay | Rattus norvegicus | 18 | cell-based format | Scientific Literature | ||
| 10. | ALA932846 | F | Antagonist activity at rat recombinant P2X7 receptor assessed as inhibition of calcium flux by FLIPR assay | Rattus norvegicus | 28 | assay format | Scientific Literature | ||
| 11. | ALA932853 | F | Antagonist activity at rat recombinant P2X7 receptor assessed as inhibition of BzATP-induced calcium flux by FLIPR assay | Rattus norvegicus | 38 | assay format | Scientific Literature | ||
| 12. | ALA982857 | F | Antagonist activity at rat recombinant P2X7 receptor assessed as inhibition of BzATP induced calcium flux by FLIPR assay | Rattus norvegicus | 23 | assay format | Scientific Literature | ||
| 13. | ALA970589 | F | Antagonist activity at rat cloned P2X7 receptor expressed in HEK293 cells assessed as inhibition of calcium flux by FLIPR assay | Rattus norvegicus | 59 | cell-based format | Scientific Literature | ||
| 14. | ALA964573 | F | Antagonist activity at P2X7R in BzATP-stimulated rat spinal cord assessed as decrease in fluorescent propidium iodide dye uptake at 1 uM | Rattus norvegicus | 6 | assay format | Scientific Literature | ||
| 15. | ALA958118 | F | Antagonist activity at rat recombinant P2X7 receptor expressed in human 1321N1 cells assessed as benzoyl-ATP-induced calcium flux by FLIPR assay | Rattus norvegicus | 35 | cell-based format | Scientific Literature | ||
| 16. | ALA1028698 | B | Activity at rat P2X7 receptor expressed in HEK cells assessed as effect on BzATP-induced ethidium uptake | Rattus norvegicus | 9 | cell-based format | Scientific Literature | ||
| 17. | ALA1048346 | F | Antagonist activity at rat recombinant P2X7 receptor expressed in human 1321N1 cells assessed as inhibition of agonist-induced calcium flux by fluorometric assay | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA1048350 | B | Binding affinity at rat P2X7 receptor | Rattus norvegicus | 1 | single protein format | Scientific Literature | ||
| 19. | ALA1103861 | B | Inhibition of rat P2X7 receptor assessed as inhibition of ethidium bromide accumulation | Rattus norvegicus | 2 | single protein format | Scientific Literature | ||
| 20. | ALA1212279 | F | Antagonist activity at rat P2X7 receptor ethidium bromide release assay | Rattus norvegicus | 2 | assay format | Scientific Literature |
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