| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA697056 | F | Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y1 receptor at 100 uM; IA is inactive | 8 | ALA1133995 | cell-based format | Scientific Literature | ||
| 2. | ALA751768 | F | The compound was evaluated for antagonist activity against phospholipase C coupled P2Y purinoceptor 1 (P2Y1) of turkey erythrocytes | Cavia porcellus | 1 | ALA1135773 | assay format | Scientific Literature | |
| 3. | ALA751769 | F | The compound was evaluated for antagonistic activity at P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coli | Cavia porcellus | 2 | ALA1135773 | assay format | Scientific Literature | |
| 4. | ALA751770 | B | Dissociation constant at P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coli | Cavia porcellus | 1 | ALA1135773 | single protein format | Scientific Literature | |
| 5. | ALA751771 | B | Dissociative constant at P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coli | Cavia porcellus | 1 | ALA1135773 | single protein format | Scientific Literature | |
| 6. | ALA751772 | F | The compound was evaluated for antagonistic activity at P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coli | Cavia porcellus | 2 | ALA1135773 | assay format | Scientific Literature | |
| 7. | ALA750154 | F | The compound was evaluated for antagonist activity against P2Y purinoceptor 1 (P2Y1) from guinea pig taenia coli | Cavia porcellus | 1 | ALA1135773 | assay format | Scientific Literature | |
| 8. | ALA750155 | B | Accumulation of inositol phosphate in 1321N1 astrocytoma cells expressing human P2Y1 purinoceptor | Homo sapiens | 13 | ALA1135410 | cell-based format | Scientific Literature | |
| 9. | ALA750156 | F | Evaluated for agonist activity against phospholipase C coupled P2Y purinoceptor 1 (P2Y1) of human erythrocytes | 3 | ALA1135773 | assay format | Scientific Literature | ||
| 10. | ALA750157 | F | Measure of Agonist Potency at human P2Y purinoceptor 1 (hP2Y1) stably expressed in 131N1 astrocytoma cell | 2 | ALA1135398 | assay format | Scientific Literature | ||
| 11. | ALA750158 | B | KB value was evaluated at the human P2Y purinoceptor 1 (P2Y1); IA menas inactive | 1 | ALA1135726 | single protein format | Scientific Literature | ||
| 12. | ALA750159 | F | Antagonistic activity against P2Y purinoceptor 1 | Homo sapiens | 13 | ALA1145892 | assay format | Scientific Literature | |
| 13. | ALA750160 | B | KB value was evaluated at the human P2Y purinoceptor 1 (P2Y1) | 1 | ALA1135726 | single protein format | Scientific Literature | ||
| 14. | ALA750161 | B | Inhibition of [3H]5 binding to P2Y purinoceptor 1 expressed in Sf9 cells | Homo sapiens | 13 | ALA1145892 | cell-based format | Scientific Literature | |
| 15. | ALA750162 | F | Agonist activity by measuring P2Y purinoceptor 1-promoted phospholipase Cactivity in human erythrocyte membranes;NE means no effect. | 1 | ALA1135410 | cell membrane format | Scientific Literature | ||
| 16. | ALA750163 | F | Agonist activity by measuring inositol phosphate accumulation in 1321N1 human astrocytoma cells stably expressing human P2Y purinoceptor 1; No effect as either agonist or antagonist at 10 uM | 4 | ALA1135410 | assay format | Scientific Literature | ||
| 17. | ALA750164 | B | pA2 value was evaluated against P2Y purinoceptor 1 | 2 | ALA1135726 | single protein format | Scientific Literature | ||
| 18. | ALA759181 | F | Evaluated for agonist activity against phospholipase C coupled P2Y purinoceptor 1 (P2Y1) of rat erythrocytes | Rattus norvegicus | 1 | ALA1135773 | assay format | Scientific Literature | |
| 19. | ALA766586 | F | Compound was measured for the antagonism of the activation of phospholipase C in mutant(F131A) human P2Y1 receptor in presence of MRS2179 (P<0.05) | 1 | ALA1131534 | assay format | Scientific Literature | ||
| 20. | ALA768341 | F | Compound was measured for the antagonism of the activation of phospholipase C in mutant(F131A) human P2Y1 receptor. | 1 | ALA1131534 | assay format | Scientific Literature |
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