| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2209112 | B | Inhibition of MLL3 using core histone as substrate preincubated for 10 mins followed by addition of [3H]SAM and incubated for 60 mins | 1 | single protein format | Scientific Literature | |||
| 2. | ALA3784088 | B | Inhibition of human MLL3 at 10 and 50 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA3821569 | B | Inhibition of MLL3 (unknown origin) at 1 to 50 uM by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA3859061 | B | Inhibition of MLL3 (unknown origin) at 50 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA4005617 | B | Inhibition of MLL3 (unknown origin) at 10 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA4005646 | B | Inhibition of MLL3 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA4017386 | B | Inhibition of MLL3 (unknown origin) H3K4 methyltransferase activity using biotinyl-H3 peptide (1 to 21 residues) and using [3H]-S adenosylmethionine as methyl donor up to 100 uM after 1 hr by scintillation counting | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA4346627 | B | Inhibition of MLL3 (unknown origin) assessed as reduction in incorporation of [3H]-labeled methyl group into biotinylated substrate using [3H-SAM] at 10 uM incubated for 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA4480237 | B | Inhibition of MLL3 (unknown origin) using biotin-labeled histone substrate assessed as residual activity at 50 uM in presence of [3H-Me]SAM by scintillation proximity assay relative to control | Homo sapiens | 24 | single protein format | Scientific Literature | ||
| 10. | ALA5030806 | B | Inhibition of MLL3 (unknown origin) at 1 to 10 uM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 11. | ALA5119837 | B | Inhibition of human recombinant N-terminal his-tagged MLL3 (4689 to 4911 residues) expressed in Escherichia coli at 10 uM using H3 as substrate by scintillation/filter assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA5119874 | B | Inhibition of human recombinant N-terminal his-tagged MLL3 (4689 to 4911 residues) expressed in Escherichia coli at 50 uM using H3 as substrate by scintillation/filter assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature |
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