# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA699705 | B | Inhibition constant (Ki) for human intestinal peptide carrier | 104 | ALA1145942 | single protein format | Scientific Literature | ||
2. | ALA699706 | B | Concentration required to inhibit the maximum [14C]Gly-Sar uptake by human Intestinal peptide transporter PepT1 in Caco-2 cells | Homo sapiens | 5 | ALA1149319 | cell-based format | Scientific Literature | |
3. | ALA699707 | B | Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]Gly-Sar uptake | Homo sapiens | 5 | ALA1149319 | cell-based format | Scientific Literature | |
4. | ALA841787 | B | Binding affinity against membrane transport protein PEPT1 in human Caco-2 cells | Homo sapiens | 118 | ALA1140305 | cell-based format | Scientific Literature | |
5. | ALA876384 | B | Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-Sar | Homo sapiens | 5 | ALA1138751 | single protein format | Scientific Literature | |
6. | ALA831529 | B | Inhibition of [14C]Gly-Sar transport by hPEPT1 in Caco-2 cell monolayers | Homo sapiens | 5 | ALA1138751 | cell-based format | Scientific Literature | |
7. | ALA829539 | B | Inhibitory concentration against [3H]glycylsarcosine uptake in HeLa cells expressing human Intestinal peptide transporter PepT1 | Homo sapiens | 14 | ALA1142674 | cell-based format | Scientific Literature | |
8. | ALA829220 | B | Relative inhibition of [3H]glycylsarcosine uptake in HeLa cells expressing human Intestinal peptide transporter PepT1 compared to BDCRB | Homo sapiens | 12 | ALA1142674 | cell-based format | Scientific Literature | |
9. | ALA829222 | B | Relative inhibition of [3H]glycylsarcosine uptake in HeLa cells expressing human Intestinal peptide transporter PepT1 compared to BDCRB; na=Not applicable | Homo sapiens | 2 | ALA1142674 | cell-based format | Scientific Literature | |
10. | ALA863210 | F | Activation of human PEPT1 expressed in MDCK cells | Homo sapiens | 80 | ALA1148644 | cell-based format | Scientific Literature | |
11. | ALA863211 | F | Activation of human PEPT1 expressed in MDCK cells relative to Gly-Sar | Homo sapiens | 79 | ALA1148644 | cell-based format | Scientific Literature | |
12. | ALA863212 | F | Ratio of %GSmax to EC50 for human PEPT1 activation | Homo sapiens | 59 | ALA1148644 | assay format | Scientific Literature | |
13. | ALA863213 | F | Binding affinity to human PEPT1 assessed as inhibition of [14C]Gly-Sar uptake in MDCK cells | Homo sapiens | 81 | ALA1148644 | cell-based format | Scientific Literature | |
14. | ALA871421 | B | Displacement of [14C]Gly-Sar from human PEPT1 in Caco-2 cells | Homo sapiens | 3 | ALA1138082 | cell-based format | Scientific Literature | |
15. | ALA896860 | B | Inhibition of [3H]GlySar uptake at human PepT1 in Caco-2 cells | Homo sapiens | 11 | ALA1148825 | cell-based format | Scientific Literature | |
16. | ALA937504 | B | Inhibition of human PEPT1-mediated [3H]GlySar uptake in CHO cells at 1 mM | Homo sapiens | 3 | ALA1144795 | cell-based format | Scientific Literature | |
17. | ALA974305 | B | Activity of human PepT1 expressed in xenopus laevis oocyte assessed as induction of inward current at 5 mM | Homo sapiens | 4 | ALA1156499 | assay format | Scientific Literature | |
18. | ALA974306 | B | Activity of human PepT1 expressed in xenopus laevis oocyte assessed as induction of inward current | Homo sapiens | 2 | ALA1156499 | assay format | Scientific Literature | |
19. | ALA1066196 | B | Inhibition of human PEPT1-mediated [3H]Gly-Sar uptake in human HeLa cells | Homo sapiens | 8 | ALA1157698 | cell-based format | Scientific Literature | |
20. | ALA1743153 | A | Substrates of transporters of clinical importance in the absorption and disposition of drugs, PEPT1 | Homo sapiens | 8 | ALA1743141 | single protein format | Scientific Literature |