| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2330198 | B | Inhibition of SUV420H2 (unknown origin) using histone H4 (1 to 24)K20Me1 as substrate after 1 hr by scintillation proximity assay in presence of [3H]-S-adenosylmethionine | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 2. | ALA3111730 | B | Inhibition of SUV420H2 (unknown origin)-mediated incorporation of methyl group from [3H]-SAM into peptide substrate up to 50 uM by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA3378211 | B | Inhibition of SUV420H2 (unknown origin) assessed as incorporation of tritium-labeled methyl group to lysine or arginine residues of peptide substrate by radioactive assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA3399139 | B | Inhibition of SUV420H2 (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 5. | ALA3399146 | B | Inhibition of SUV420H2 (unknown origin) at 10 uM by HMT assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA3592399 | B | Inhibition of SUV420H2 (unknown origin) at 1 uM after 1 hr by filter-based assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA3784103 | B | Inhibition of human SUV420H2 at 10 and 50 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA3821907 | B | Inhibition of SUV420H2 (unknown origin) at 1 to 50 uM by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA3859076 | B | Inhibition of SUV420H2 (unknown origin) at 50 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4005615 | B | Inhibition of SUV420H2 (unknown origin) at 10 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4005644 | B | Inhibition of SUV420H2 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4346629 | B | Inhibition of SUV420H2 (unknown origin) assessed as reduction in incorporation of [3H]-labeled methyl group into biotinylated substrate using [3H-SAM] at 10 uM incubated for 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4376158 | B | Inhibition of SUV420H2 (unknown origin) at 1 uM using biotin-labeled peptide as substrate and [3H]-SAM measured after 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA4376161 | B | Inhibition of SUV420H2 in human MCF7 cells assessed as decrease in H4K20me3 level up to 50 uM measured after 2 days by immunoblot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA4377314 | B | Inhibition of human SUV420H2 up to 50 uM using Biot-H4K20me1 as substrate and in presence of [3H]-SAM incubated for 1 hr by scintillation proximity assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA4480251 | B | Inhibition of SUV420H2 (unknown origin) using biotin-labeled histone substrate assessed as residual activity at 50 uM in presence of [3H-Me]SAM by scintillation proximity assay relative to control | Homo sapiens | 24 | single protein format | Scientific Literature | ||
| 17. | ALA5030784 | B | Inhibition of SUV420H2 (unknown origin) at 1 to 10 uM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 18. | ALA5210095 | B | Affinity Phenotypic Cellular interaction (Western Blot (decrease in di-methylation of H4K20me in U20S cells)) EUB0000193b SUV420H2 | Homo sapiens | 1 | cell-based format | Literature data from EUbOPEN Chemogenomic Library | ||
| 19. | ALA5210588 | B | Affinity Biochemical interaction (Scintillation proximity assay (SPA)) EUB0000193b SUV420H2 | Homo sapiens | 1 | single protein format | Literature data from EUbOPEN Chemogenomic Library | ||
| 20. | ALA5213733 | B | Selectivity interaction (Protein methyltransferase panel (activity assay)) EUB0000211b SUV420H2 | Homo sapiens | 1 | single protein format | Literature data from EUbOPEN Chemogenomic Library |
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