| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA621841 | F | Compound tested for relative response using 1 uM ACh as agonist against AChM1 receptor. | 1 | assay format | Scientific Literature | |||
| 2. | ALA714427 | B | Ability to displace [3H]pirenzepine (PZ) from M1 receptor in rat cortex homogenate | 4 | tissue-based format | Scientific Literature | |||
| 3. | ALA714428 | B | Affinity constant against Muscarinic acetylcholine receptor M1 of rat cerebral cortex. | 1 | tissue-based format | Scientific Literature | |||
| 4. | ALA714429 | B | Affinity constant to Muscarinic acetylcholine receptor M1 of rat cerebral cortex | 1 | tissue-based format | Scientific Literature | |||
| 5. | ALA714430 | F | Compound was measured for percentage of intrinsic activity against M1 muscarinic receptor, by stimulation of phosphatidylinositol (PI) hydrolysis in rat hippocampal slices | 4 | tissue-based format | Scientific Literature | |||
| 6. | ALA877252 | B | Pseudo hill coefficient at M1 receptor | 1 | single protein format | Scientific Literature | |||
| 7. | ALA711165 | B | Pseudo hill coefficient at Muscarinic acetylcholine receptor M1 | 2 | single protein format | Scientific Literature | |||
| 8. | ALA711166 | B | Binding affinity at [3H]PZ radiolabeled muscarinic M1 receptor in rat cortex. | 18 | tissue-based format | Scientific Literature | |||
| 9. | ALA858414 | B | Affinity constant measured against M1 muscarinic receptor in rat cortex | 4 | assay format | Scientific Literature | |||
| 10. | ALA711327 | B | The binding affinity was measured on muscarine M1 receptor using [3H]- pirenzepine as radioligand. | 2 | single protein format | Scientific Literature | |||
| 11. | ALA719078 | B | Compound is tested for displacement of [3H]pirenzepine at Metabotropic glutamate receptor 1 in Rat brain homogenate. | 8 | tissue-based format | Scientific Literature | |||
| 12. | ALA747765 | B | Affinity for muscarinic receptor M1 in rat brain was measured by inhibition of [3H](R)-quinuclidinyl benzilate (QNB) binding | 3 | tissue-based format | Scientific Literature | |||
| 13. | ALA747775 | B | Binding affinity against Muscarinic receptor M1 in rat brain using [3H]-PZ (pirenzepine) radioligand at a concentration of 1 nM | 5 | tissue-based format | Scientific Literature | |||
| 14. | ALA878551 | B | The compound was tested in vitro for binding activity against M1 muscarinic receptor in homogenates of the cerebral cortex of rat using [3H]pirenzepine as radioligand | 3 | tissue-based format | Scientific Literature | |||
| 15. | ALA748058 | B | Inhibition of binding of [3H]quinuclidinyl benzilate to Muscarinic acetylcholine receptor M1 in rat brain cortex at 10e-5 M of compound concentration; Less active | 3 | tissue-based format | Scientific Literature | |||
| 16. | ALA748059 | B | Inhibition of binding of [3H]quinuclidinyl benzilate to Muscarinic acetylcholine receptor M1 in rat brain cortex at 10e-5 M of compound concentration; Less active | 7 | tissue-based format | Scientific Literature | |||
| 17. | ALA748060 | F | Compound was tested in vitro for depolarizing response on the rat superior cervical ganglion (mediated by Muscarinic M1 receptor | 1 | tissue-based format | Scientific Literature | |||
| 18. | ALA748061 | F | Compound was tested in vitro for depolarizing response on the rat superior cervical ganglion (mediated by Muscarinic M1 receptor) | 1 | tissue-based format | Scientific Literature | |||
| 19. | ALA748215 | F | Compound was tested in vitro for depolarizing response on the rat superior cervical ganglion (mediated by muscarinic acetylcholine receptor M1) | 1 | tissue-based format | Scientific Literature | |||
| 20. | ALA748216 | F | Inhibitory activity against stimulation of [3H]inositol monophosphate accumulation in [3H]inositol-labelled CHO transfected cells mediated by Muscarinic acetylcholine receptor M1 | 4 | cell-based format | Scientific Literature |
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