# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA935756 | B | Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in HEK293 cells | Mus musculus | 9 | ALA1145629 | cell-based format | Scientific Literature | |
2. | ALA923562 | B | Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarbox-amidoadenosine from mouse recombinant adenosine A2A receptor expressed in HEK293 at 100 uM | Mus musculus | 14 | ALA1145629 | cell-based format | Scientific Literature | |
3. | ALA2067574 | B | Displacement of [3H]I-AB-MECA from mouse adenosine A2A receptor expressed in HEK293 cells at 10 uM after 60 mins by liquid scintillation counting | Mus musculus | 11 | ALA2062514 | cell-based format | Scientific Literature | |
4. | ALA2404652 | B | Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5'-N-ethylcarboxamidoadenosine from mouse adenosine A2A receptor expressed in HEK293 cell membranes at 10 uM after 60 mins by liquid scintillation counting analysis relative to control | Mus musculus | 12 | ALA2401698 | cell-based format | Scientific Literature | |
5. | ALA3095019 | F | Antagonist activity at adenosine A2A receptor in C57/BL6 mouse lymphocytes assessed as inhibition of CGS-21680-mediated cAMP accumulation after 15 mins by ELISA | Mus musculus | 1 | ALA3091430 | cell-based format | Scientific Literature | |
6. | ALA3095020 | F | Antagonist activity at adenosine A2A receptor in C57/BL6 mouse lymphocytes assessed as inhibition of CGS-21680-mediated cAMP accumulation at 0.5 to 10 uM after 15 mins by ELISA | Mus musculus | 2 | ALA3091430 | cell-based format | Scientific Literature | |
7. | ALA3413618 | B | Displacement of [3H]CGS21680 from mouse A2A adenosine receptor expressed in HEK293 cells at 10 uM after 60 mins by liquid scintillation counting | Mus musculus | 7 | ALA3407461 | cell-based format | Scientific Literature | |
8. | ALA4262951 | B | Displacement of [3H]ZM241385 from recombinant mouse adenosine receptor A2A expressed in HEK293 cell membranes after 1 hr by FACS analysis | Mus musculus | 4 | ALA4261547 | cell-based format | Scientific Literature | |
9. | ALA4346856 | B | Displacement of [3H]MSX-2 from recombinant mouse A2A adenosine receptor expressed in CHO cell membranes measured after 60 mins by liquid scintillation counting method | Mus musculus | 2 | ALA4346653 | cell-based format | Scientific Literature | |
10. | ALA4369166 | A | Displacement of [3H]ZM241385 from mouse A2A receptor at 10 uM | Mus musculus | 1 | ALA4368860 | single protein format | Scientific Literature | |
11. | ALA4369924 | B | Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from mouse A2A adenosine receptor expressed in HEK293 cell membranes at 10 uM after 60 mins by scintillation proximity assay relative to adenosine 5-N-ethyluronamide | Mus musculus | 7 | ALA4368904 | cell-based format | Scientific Literature | |
12. | ALA4369926 | B | Displacement of [3H]2-[p-(2-carboxyethyl)phenylethylamino]-5-N-ethylcarboxamidoadenosine from mouse A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by scintillation proximity assay | Mus musculus | 4 | ALA4368904 | cell-based format | Scientific Literature | |
13. | ALA4423031 | B | Antagonist activity at recombinant mouse A2A adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assay | Mus musculus | 1 | ALA4422615 | cell-based format | Scientific Literature | |
14. | ALA4701038 | B | Antagonist activity at adenosine 2A receptor in BALB/c mouse T cells assessed as reduction in CGS-21680-induced suppression of IL-2 secretion incubated for 24 hrs by ELISA | Mus musculus | 1 | ALA4699449 | cell-based format | Scientific Literature | |
15. | ALA4701039 | B | Antagonist activity at adenosine 2A receptor in BALB/c mouse T cells assessed as reduction in CGS-21680-induced suppression of IFN-gamma secretion incubated for 24 hrs by ELISA | Mus musculus | 1 | ALA4699449 | cell-based format | Scientific Literature | |
16. | ALA4731040 | B | Displacement of [3H]CGS21680 from mouse A2A receptor expressed in HEK293 cells at 10 uM by radio ligand binding assay relative to control | Mus musculus | 5 | ALA4725439 | cell-based format | Scientific Literature | |
17. | ALA5042370 | B | Displacement of [3H] ZM241385 from mouse adenosine A2A receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assay | Mus musculus | 1 | ALA5038675 | cell-based format | Scientific Literature | |
18. | ALA5042374 | B | Displacement of [3H] ZM241385 from mouse adenosine A2A receptor expressed in HEK293 cells at 10 uM incubated for 60 mins by radioligand binding assay | Mus musculus | 3 | ALA5038675 | cell-based format | Scientific Literature | |
19. | ALA5155954 | B | Binding affinity to mouse adenosine A2A receptor expressed in human HEK293 cell membrane by radioligand inhibition assay | Mus musculus | 1 | ALA5154659 | cell membrane format | Scientific Literature |