# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3429882 | Binding | Inhibition of human IKKalpha | Homo sapiens | 1 | ALA3425429 | single protein format | Scientific Literature | |
2. | ALA3428314 | Binding | Inhibition of human IKKa/CHUK using KKKKERLLDDRHDSGLDSMKDEE peptide substrate at 1 uM by 33P Hotspot assay | Homo sapiens | 1 | ALA3425491 | single protein format | Scientific Literature | |
3. | ALA3630662 | Binding | Inhibition of IKK-alpha (unknown origin) assessed as remaining activity at 10 uM by high-throughput assay relative to control | Homo sapiens | 1 | ALA3627674 | single protein format | Scientific Literature | |
4. | ALA3631254 | Binding | Inhibition of IKKalpha (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
5. | ALA3737506 | Binding | Inhibition of IKKalpha (unknown origin) at 1 uM by selectscreen kinase profiling assay in presence of ATP | Homo sapiens | 1 | ALA3734692 | single protein format | Scientific Literature | |
6. | ALA3744692 | Binding | Inhibition of TNF-alpha-induced IKK-alpha phosphorylation in human MDA-MB-231 cells at Ser176 residue at 5 and 10 uM pretreated for 30 mins followed by addition of TNF-alpha for 1 hr by immunoblot analysis | Homo sapiens | 1 | ALA3739305 | cell-based format | Scientific Literature | |
7. | ALA3751250 | Binding | Inhibition of IKK alpha (unknown origin) at 1 uM | Homo sapiens | 1 | ALA3745631 | single protein format | Scientific Literature | |
8. | ALA3748216 | Binding | Inhibition of human IKKalpha using [KKKKERLLDDRHDSGLDSMKDEE] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
9. | ALA3762887 | Binding | Inhibition of IKKalpha (unknown origin) at 100 nM | Homo sapiens | 2 | ALA3758169 | single protein format | Scientific Literature | |
10. | ALA3767310 | Binding | Inhibition of IKKalpha (unknown origin) at 10 uM | Homo sapiens | 1 | ALA3763027 | single protein format | Scientific Literature | |
11. | ALA3771579 | Binding | Inhibition of human recombinant IKKalpha assessed as residual activity at 10 uM after 1 hr by qPCR analysis relative to control | Homo sapiens | 1 | ALA3769377 | single protein format | Scientific Literature | |
12. | ALA3776218 | Binding | Inhibition of N-terminal His6-tagged recombinant human IKKalpha expressed in baculovirus infected insect Sf9 cells assessed as remaining activity at 1 uM relative to control | Homo sapiens | 3 | ALA3774357 | cell-based format | Scientific Literature | |
13. | ALA3782177 | Binding | Inhibition of partial length human IKKalpha expressed in mammalian system at 1 uM | Homo sapiens | 1 | ALA3779767 | assay format | Scientific Literature | |
14. | ALA3787881 | Binding | Inhibition of human recombinant His tagged IKK1 expressed in baculovirus at 10 uM after 60 mins by Adapta assay | Homo sapiens | 13 | ALA3785011 | assay format | Scientific Literature | |
15. | ALA3812178 | Binding | Inhibition of His-tagged full length human recombinant IKKalpha expressed in baculovirus using Fluorescein-IKK as substrate at 100 nM | Homo sapiens | 1 | ALA3808348 | assay format | Scientific Literature | |
16. | ALA3812433 | Binding | Inhibition of full length human IKK-alpha assessed as enzyme activity at 10 uM by KINOMEScan assay | Homo sapiens | 1 | ALA3808372 | single protein format | Scientific Literature | |
17. | ALA3816701 | Binding | Inhibition of human IKKalpha at 1 uM using [KKKKERLLDDRHDSGLDSMKDEE] as substrate | Homo sapiens | 1 | ALA3813650 | single protein format | Scientific Literature | |
18. | ALA3817193 | Binding | Inhibition of full length recombinant human His-tagged IKK-alpha expressed in baculovirus expression system at 1 uM relative to control | Homo sapiens | 1 | ALA3813614 | assay format | Scientific Literature | |
19. | ALA3820338 | Binding | Inhibition of full length recombinant human N-terminal GST-tagged IKKalpha expressed in baculovirus infected Sf21 cells at 1 uM by radiometric assay relative to control | Homo sapiens | 2 | ALA3817791 | cell-based format | Scientific Literature | |
20. | ALA3826036 | Binding | Inhibition of His-tagged full-length human IKKalpha expressed in baculovirus system at 100 nM by adapta assay | Homo sapiens | 1 | ALA3822377 | assay format | Scientific Literature |