| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2382489 | B | Inhibition of PARP7 (unknown origin) at 10 uM relative to control | Homo sapiens | 2 | ALA2380224 | single protein format | Scientific Literature | |
| 2. | ALA3242399 | B | Inhibition of recombinant human PARP-7 at 10 uM relative to control | Homo sapiens | 1 | ALA3232733 | single protein format | Scientific Literature | |
| 3. | ALA3382574 | B | Inhibition of human recombinant PARP7 at 10 uM incubated for 1 hr using using NAD+, biotinylated NAD+ and activated DNA by luminescence based assay | Homo sapiens | 1 | ALA3351316 | single protein format | Scientific Literature | |
| 4. | ALA3382584 | B | Inhibition of human recombinant PARP7 at 100 uM incubated for 1 hr using using NAD+, biotinylated NAD+ and activated DNA by luminescence based assay | Homo sapiens | 1 | ALA3351316 | single protein format | Scientific Literature | |
| 5. | ALA4311847 | B | Inhibition of human PARP7 assessed as reduction in MARylation of SRPK2 substrate after 60 mins in presence of 6-a-NAD+ by chemifluorescence assay | Homo sapiens | 1 | ALA4308918 | single protein format | Scientific Literature | |
| 6. | ALA4322266 | B | Inhibition of N-terminal FLAG-tagged recombinant human PARP7 (400 to 657 residues) expressed in Baculovirus infected Sf9 cells using biotinylated substrate after 1 hr by chemiluminescence method | Homo sapiens | 1 | ALA4321794 | cell-based format | Scientific Literature | |
| 7. | ALA4678527 | B | Inhibition of PARP-7 (unknown origin) pre-incubated for 30 mins before addition of activated DNA and NAD by chemiluminescent assay | Homo sapiens | 1 | ALA4673340 | single protein format | Scientific Literature | |
| 8. | ALA4701309 | B | Inhibition of N-terminal FLAG-tagged human PARP7 (400 to 657 residues) expressed in baculovirus infected Sf9 cells assessed as reduction in NAD+-dependent ADP ribosylation using histone as substrate at 10 uM incubated for 1 hr in presence of biotinylated NAD+ and activated DNA by chemiluminescence based microplate reader assay relative to control | Homo sapiens | 2 | ALA4699460 | cell-based format | Scientific Literature | |
| 9. | ALA5108309 | B | Inhibition of N-terminal His-tagged full length human PARP7 expressed in Escherichia coli BL21 (DE3) at 10 uM preincubated with 6-a-NAD+ for 5 to 10 mins followed by enzyme addition and measured after 60 mins using NAD+ as substrate byHRP based chemiluminescence assay | Homo sapiens | 6 | ALA5107944 | assay format | Scientific Literature | |
| 10. | ALA5123576 | B | Displacement of fluorescent labeled RBN011198 from human NanoLuc-tagged full-length PARP7 expressed in HEK293T cells using NanoGlo substrate incubated for 2 hrs by NanoBRET assay | Homo sapiens | 1 | ALA5120855 | cell-based format | Scientific Literature | |
| 11. | ALA5123673 | B | Inhibition of PARP-7 (unknown origin) | Homo sapiens | 1 | ALA5120857 | single protein format | Scientific Literature | |
| 12. | ALA5124502 | B | Inhibition of PARP7 (unknown origin) | Homo sapiens | 2 | ALA5120882 | single protein format | Scientific Literature | |
| 13. | ALA5124507 | B | Binding affinity to PARP7 (unknown origin) assessed as dissociation constant | Homo sapiens | 1 | ALA5120882 | single protein format | Scientific Literature | |
| 14. | ALA5131328 | B | Inhibition of PARP7 (unknown origin) by HTRF assay | Homo sapiens | 12 | ALA5126675 | single protein format | Scientific Literature | |
| 15. | ALA5152045 | B | Binding affinity to PARP7 (unknown origin) assessed as apparent dissociation constant | Homo sapiens | 6 | ALA5150005 | single protein format | Scientific Literature | |
| 16. | ALA5228293 | B | Inhibition of N-terminal FLAG-tagged human recombinant PARP7 (400 to 657 residues) expressed in Sf9 insect cells by chemiluminescence assay | Homo sapiens | 1 | ALA5226325 | cell-based format | Scientific Literature |
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