# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2424428 | B | Inhibition of NEK8 in human PC3 cell lysates at 10 uM using desthiobiotin-tagged ATP probe AX9989 followed by trypsinization by LC/MS analysis | Homo sapiens | 12 | single protein format | Scientific Literature | ||
2. | ALA4034428 | B | Inhibition of NEK8 Lysine 2 labelling site (unknown origin) at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
3. | ALA4045779 | B | Inhibition of NEK8 conserved Lys2 (DLKTQNILLDK) in human PBMC at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
4. | ALA4046020 | B | Inhibition of NEK8 conserved Lys2 (DLKTQNILLDK) in human PBMC at 0.1 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
5. | ALA4118429 | B | Inhibition of NEK8 in human SKCO1 cells at 1 uM after 4 hrs using biotin labeled DLKTQNILLDK probe by mass-spectrometric analysis relative to control | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
6. | ALA4327802 | B | Inhibition of human NEK8 assessed as residual activity at 1 uM using casein as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
7. | ALA4328166 | B | Inhibition of human NEK8 assessed as residual activity at 100 uM using casein as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
8. | ALA4328530 | B | Inhibition of human NEK8 using casein as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
9. | ALA4366514 | B | Inhibition of human NEK8 at 100 nM using casein as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
10. | ALA4405487 | B | Inhibition of NEK8 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
11. | ALA4674272 | B | Inhibition of human NEK8 using casein as substrate assessed as residual activity at 1 uM by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | single protein format | Scientific Literature | ||
12. | ALA4720626 | B | Inhibition of human NEK8 using casein as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
13. | ALA4720972 | B | Inhibition of human NEK8 assessed as residual activity using casein as substrate at 1 uM by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
14. | ALA4804448 | B | Inhibition of NEK8 in human NCI-H929 cells by mass spectroscopic analysis | Homo sapiens | 6 | cell-based format | Patent Bioactivity Data | ||
15. | ALA4804630 | B | Inhibition of NEK8 in human NCI-H929 cells at 10 uM by mass spectroscopic analysis relative to control | Homo sapiens | 6 | cell-based format | Patent Bioactivity Data | ||
16. | ALA4884794 | B | Nek8(NEK8LGRI) Takeda global kinase panel | Homo sapiens | 1 | single protein format | Donated Chemical Probes - SGC Frankfurt | ||
17. | ALA4885085 | B | Nek8(NEK8LGRI) Takeda global kinase panel | Homo sapiens | 1 | single protein format | Donated Chemical Probes - SGC Frankfurt | ||
18. | ALA4887296 | B | NEK8 Invitrogen Lab (UK) kinase screen (BI) | Homo sapiens | 1 | single protein format | Donated Chemical Probes - SGC Frankfurt | ||
19. | ALA5058299 | B | Inhibition of NEK8 (unknown origin) at 1 uM | Homo sapiens | 1 | single protein format | Scientific Literature |