# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2427608 | B | Inhibition of KDM5A (unknown origin) using H3K4me3 peptide and 2-oxoglutarate as substrate after 1 hr by FDH-coupled assay | Homo sapiens | 12 | ALA2424657 | single protein format | Scientific Literature | |
2. | ALA2429070 | B | Inhibition of JARID1A (unknown origin) after 30 mins by AlphaScreen assay | Homo sapiens | 56 | ALA2424619 | single protein format | Scientific Literature | |
3. | ALA3136678 | B | Inhibition of GST-tagged Jarid1A (unknown origin) using H3K4Me3 as substrate incubated for 30 mins at room temperature followed by incubation under dark condition for 30 mins by AlphaScreen assay | Homo sapiens | 25 | ALA3132809 | single protein format | Scientific Literature | |
4. | ALA3591676 | B | Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay | Homo sapiens | 17 | ALA3588787 | single protein format | Scientific Literature | |
5. | ALA3591680 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K9me3/H3 ratio at 300 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
6. | ALA3591681 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K4me3/H3 ratio at 100 uM after 24 hrs by Western blot analysis | Homo sapiens | 4 | ALA3588787 | cell-based format | Scientific Literature | |
7. | ALA3591682 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K4me3/H3 ratio at 300 uM after 24 hrs by Western blot analysis | Homo sapiens | 4 | ALA3588787 | cell-based format | Scientific Literature | |
8. | ALA3591683 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as increase in accumulation of H3K4me3 after 24 hrs by Western blot analysis | Homo sapiens | 2 | ALA3588787 | cell-based format | Scientific Literature | |
9. | ALA3591684 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K4me3/H3 ratio at 30 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
10. | ALA3591685 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K4me3/H3 ratio at 10 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
11. | ALA3591686 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K9me3/H3 ratio at 100 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
12. | ALA3591687 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K9me3/H3 ratio at 30 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
13. | ALA3591688 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K9me3/H3 ratio at 10 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
14. | ALA3591816 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K27me3/H3 ratio at 300 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
15. | ALA3591817 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K27me3/H3 ratio at 100 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
16. | ALA3591818 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K27me3/H3 ratio at 30 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
17. | ALA3591819 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K27me3/H3 ratio at 10 uM after 24 hrs by Western blot analysis | Homo sapiens | 1 | ALA3588787 | cell-based format | Scientific Literature | |
18. | ALA3624712 | B | Inhibition of KDM5A (unknown origin) by alpha screen assay | Homo sapiens | 1 | ALA3621091 | single protein format | Scientific Literature | |
19. | ALA3776332 | B | Inhibition of KDM5A (1 to 797 residues) (unknown origin) expressed in insect sf21 cells using ARTK(Me3)QTARKSTGGKAPRK peptide/ 100 uM alpha-ketoglutarate as substrate/cofactor incubated for 45 mins by MALDI assay | Homo sapiens | 6 | ALA3774347 | cell-based format | Scientific Literature | |
20. | ALA3777864 | B | Inhibition of JARID1A (unknown origin) using H3K4me3 peptide substrate preincubated for 5 mins followed by substrate addition by MALDI-TOF mass spectrometric analysis | Homo sapiens | 8 | ALA3774333 | single protein format | Scientific Literature |