# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA941813 | B | Inhibition of TAK1-TAB1 | Homo sapiens | 1 | ALA1140564 | assay format | Scientific Literature | |
2. | ALA1105931 | B | Inhibition of TAK1/TAB1 at 5 uM | 1 | ALA1154316 | protein complex format | Scientific Literature | ||
3. | ALA1763403 | B | Competitive inhibition of recombinant TAK1-TAB1 assessed as [33P]gamma-ATP incorporation into substrate histone H1 peptide by filter plate assay | 23 | ALA1759936 | protein complex format | Scientific Literature | ||
4. | ALA1763404 | B | Competitive inhibition of recombinant TAK1-TAB1 assessed as [33P]gamma-ATP incorporation into substrate histone H1 peptide at 10 uM by filter plate assay | 24 | ALA1759936 | protein complex format | Scientific Literature | ||
5. | ALA1931563 | B | Inhibition of TAK1-TAB1 | 2 | ALA1926590 | protein complex format | Scientific Literature | ||
6. | ALA2015521 | B | Inhibition of TAK1-TAB1 at 10 uM | 1 | ALA2010722 | protein complex format | Scientific Literature | ||
7. | ALA2404317 | B | Inhibition of TAK1/TAB1 (unknown origin) at 10 uM relative to control | Homo sapiens | 1 | ALA2401733 | protein complex format | Scientific Literature | |
8. | ALA2412856 | B | Inhibition of truncated TAK1-TAB1(unknown origin) using MKK7 as substrate by ALPHAScreen assay in presence of ATP | Homo sapiens | 59 | ALA2407040 | protein complex format | Scientific Literature | |
9. | ALA2410824 | B | Inhibition of TAK1-TAB1 (unknown origin) by alphascreen assay in presence of ATP | Homo sapiens | 25 | ALA2407065 | protein complex format | Scientific Literature | |
10. | ALA3124032 | B | Inhibition of TAK1/TAB1 (unknown origin) at 0.1 uM relative to control | Homo sapiens | 1 | ALA3120096 | protein complex format | Scientific Literature | |
11. | ALA3240754 | B | Inhibition of human TAK1-TAB1 assessed as enzyme activity at 1 uM relative to control | Homo sapiens | 1 | ALA3232845 | protein complex format | Scientific Literature | |
12. | ALA3378753 | B | Inhibition of Tak1-TAB1 (unknown origin) assessed as enzyme activity by Kinase-Glo Plus luminescence kinase assay | Homo sapiens | 14 | ALA3352065 | protein complex format | Scientific Literature | |
13. | ALA3631696 | B | Inhibition of TAK1-TAB1 (unknown origin) at 1 uM by FRET method | Homo sapiens | 1 | ALA3627690 | protein complex format | Scientific Literature | |
14. | ALA3761203 | B | Inhibition of TAK1-TAB1 (unknown origin) at 100 nM | Homo sapiens | 2 | ALA3758169 | protein complex format | Scientific Literature | |
15. | ALA3807330 | B | Inhibition of full length human recombinant His-tagged TAK1-TAB1 (437 to 504 residues) expressed in baculovirus expression system at 1 uM by LanthaScreen assay relative to control | Homo sapiens | 2 | ALA3804775 | assay format | Scientific Literature | |
16. | ALA3880356 | B | Inhibition of kinase tracer-236 binding to full length recombinant human His-tagged TAK1-TAB1 expressed in baculovirus by FRET assay | Homo sapiens | 36 | ALA3879912 | assay format | Patent Bioactivity Data | |
17. | ALA4120141 | B | Inhibition of recombinant full length His-tagged human TAK1-TAB1 (437 to 504 residues) expressed in baculovirus expression system at 1 uM by FRET assay relative to control | Homo sapiens | 2 | ALA4118097 | assay format | Scientific Literature | |
18. | ALA4178172 | B | Inhibition of human TAK1 (1 to 303 residues)/TAB1 (437 to 504 residues) assessed as residual activity at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | protein complex format | Scientific Literature | |
19. | ALA4178181 | B | Inhibition of human TAK1 (1 to 303 residues)/TAB1 (437 to 504 residues) at 500 nM in presence of 33P-ATP by filter binding assay relative to control | Homo sapiens | 1 | ALA4177526 | protein complex format | Scientific Literature | |
20. | ALA4331207 | B | Inhibition of TAK1/TAB1 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA4330074 | protein complex format | Scientific Literature |