| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3089617 | B | Displacement of fluorescein-labeled MS239 from recombinant human BPTF after 1 hr by fluorescence anisotropy assay | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 2. | ALA3383407 | B | Inhibition of human BPTF by BROMOscan assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA3591388 | B | Binding affinity to BPTF in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assay | Homo sapiens | 3 | cell-based format | Scientific Literature | ||
| 4. | ALA3743458 | B | Binding affinity to human FALZ assessed as change in melting temperature at 10 uM by differential scanning fluorimetry | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA3773269 | B | Binding affinity to biotinylated FALZ (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 6. | ALA3777035 | B | Inhibition of recombinant human FALZ isoform 1 expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA3790877 | B | Binding affinity to BPTF (unknown origin) by isothermal titration calorimetric analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA3864407 | B | Displacement of biotinylated ligand from recombinant His-tagged BPTF (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 9. | ALA4012422 | B | Inhibition of FALZ (unknown origin) at 100 uM using acetylated lysine as substrate relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA4012426 | B | Inhibition of FALZ (unknown origin) at 50 uM using acetylated lysine as substrate relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA4016227 | B | Binding affinity to 5FW-labeled BPTF (unknown origin) up to 500 uM by PrOF NMR spectroscopic analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA4016245 | B | Binding affinity to 5FW-labeled BPTF (unknown origin) by PrOF NMR spectroscopic analysis | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4047549 | B | Inhibition of human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system assessed as residual activity at 500 nM relative to control by BROMOscan assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA4051566 | B | Inhibition of FALZ (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO Orange-dye based fluorescence thermal shift assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA4053075 | B | Inhibition of human His tagged FALZ incubated for 30 mins followed by addition of biotinylated peptide and further incubation for 30 mins measured by AlphaScreen assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA4058607 | B | Displacement of biotinylated histone H3K14 peptide ligand from recombinant His-tagged BPTF (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 17. | ALA4130868 | B | Inhibition of human partial length FALZ (S2791 to H2911 residues) expressed in Escherichia coli BL21 assessed as residual activity at 1 uM after 1 hr by qPCR method relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA4151036 | B | Binding affinity to human FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOScan assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA4185458 | B | Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA4186431 | B | Binding affinity to human partial length FALZ (S2791 to H2911 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 1 | assay format | Scientific Literature |
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