# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3089618 | B | Displacement of fluorescein-labeled MS226 from recombinant human BRD7 after 1 hr by fluorescence anisotropy assay | Homo sapiens | 4 | ALA3085768 | single protein format | Scientific Literature | |
2. | ALA3383415 | B | Inhibition of human BRD7 by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
3. | ALA3591392 | B | Binding affinity to BRD7 in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assay | Homo sapiens | 2 | ALA3588744 | cell-based format | Scientific Literature | |
4. | ALA3743241 | B | Binding affinity to human BRD7 by isothermal titration calorimetry | Homo sapiens | 1 | ALA3739345 | single protein format | Scientific Literature | |
5. | ALA3743450 | B | Binding affinity to human BRD7 assessed as change in melting temperature at 10 uM by differential scanning fluorimetry | Homo sapiens | 1 | ALA3739345 | single protein format | Scientific Literature | |
6. | ALA3773117 | B | Binding affinity to biotinylated BRD7 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
7. | ALA3771485 | B | Binding affinity to partial length human BRD7 by BROMOscan assay | Homo sapiens | 1 | ALA3769376 | single protein format | Scientific Literature | |
8. | ALA3777028 | B | Inhibition of recombinant human BRD7 expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
9. | ALA3778556 | B | Binding affinity to recombinant human BRD7 by differential scanning fluorimetry | Homo sapiens | 1 | ALA3774375 | single protein format | Scientific Literature | |
10. | ALA3825267 | B | Binding affinity to human BRD7 assessed as thermal shift difference at 10 uM by DSF analysis | Homo sapiens | 2 | ALA3822369 | single protein format | Scientific Literature | |
11. | ALA3826478 | B | Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen assay | Homo sapiens | 13 | ALA3822369 | assay format | Scientific Literature | |
12. | ALA3826486 | B | Inhibition of human BRD7 by VP-ITC method | Homo sapiens | 1 | ALA3822369 | single protein format | Scientific Literature | |
13. | ALA3826491 | B | Binding affinity to human BRD7 expressed in Escherichia coli L21(DE3)-R3-pRARE2 cells by VP-ITC method | Homo sapiens | 2 | ALA3822369 | cell-based format | Scientific Literature | |
14. | ALA3826492 | B | Binding affinity to human BRD7 by BROMOScan analysis | Homo sapiens | 2 | ALA3822369 | single protein format | Scientific Literature | |
15. | ALA3826493 | B | Inhibition of human BRD7 measured after mins by AlphaScreen assay | Homo sapiens | 2 | ALA3822369 | single protein format | Scientific Literature | |
16. | ALA3826013 | B | Binding affinity to human BRD7 by ITC analysis | Homo sapiens | 1 | ALA3822393 | single protein format | Scientific Literature | |
17. | ALA4012424 | B | Inhibition of BRD7 (unknown origin) at 100 uM using acetylated lysine as substrate relative to control | Homo sapiens | 1 | ALA4011609 | single protein format | Scientific Literature | |
18. | ALA4012428 | B | Inhibition of BRD7 (unknown origin) at 50 uM using acetylated lysine as substrate relative to control | Homo sapiens | 1 | ALA4011609 | single protein format | Scientific Literature | |
19. | ALA4020260 | B | Binding affinity to human BRD7 (L125 to R254 residues) expressed in mammalian expression system by BROMOscan assay | Homo sapiens | 1 | ALA4017535 | assay format | Scientific Literature | |
20. | ALA4030900 | B | Inhibition of human BRD7 (125 to 254 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assay | Homo sapiens | 1 | ALA4028852 | assay format | Scientific Literature |