| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3111496 | B | Binding affinity to BAZ2A bromodomain (unknown origin) assessed as change in melting temperature at 10 uM by differential scanning fluorimetric analysis | Homo sapiens | 35 | ALA3108763 | single protein format | Scientific Literature | |
| 2. | ALA3383405 | B | Inhibition of human BAZ2A by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
| 3. | ALA3419224 | B | Inhibition of BAZ2A (unknown origin) after 30 mins by AlphaScreen assay | Homo sapiens | 12 | ALA3414510 | single protein format | Scientific Literature | |
| 4. | ALA3419226 | B | Binding affinity to BAZ2A (unknown origin) by isothermal titration calorimetric analysis | Homo sapiens | 1 | ALA3414510 | single protein format | Scientific Literature | |
| 5. | ALA3419228 | B | Binding affinity to BAZ2A (unknown origin) assessed as thermal shift at 10 uM by Real-Time PCR analysis | Homo sapiens | 1 | ALA3414510 | single protein format | Scientific Literature | |
| 6. | ALA3419237 | B | Inhibition of N-terminal eGFP-tagged full-length BAZ2A (unknown origin) transfected in human U2OS cells assessed as reduction of protein recovery half time at 1 uM after 24 hrs by FRAP assay in presence of histone deacetylase inhibitor SAHA relative to control | Homo sapiens | 1 | ALA3414510 | cell-based format | Scientific Literature | |
| 7. | ALA3591386 | B | Binding affinity to BAZ2A in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assay | Homo sapiens | 3 | ALA3588744 | cell-based format | Scientific Literature | |
| 8. | ALA3743454 | B | Binding affinity to human BAZ2A at 10 uM by differential scanning fluorimetry | Homo sapiens | 1 | ALA3739345 | single protein format | Scientific Literature | |
| 9. | ALA3743461 | B | Binding affinity to BAZ2A (unknown origin) | Homo sapiens | 1 | ALA3739345 | single protein format | Scientific Literature | |
| 10. | ALA3772735 | B | Inhibition of recombinant His6-TEV fused human BAZ2A expressed in Escherichia coli incubated for 30 mins in presence of biotinylated peptide by alpha screen assay | Homo sapiens | 21 | ALA3769341 | assay format | Scientific Literature | |
| 11. | ALA3772740 | B | Binding affinity to recombinant His6-TEV fused human BAZ2A expressed in Escherichia coli by isothermal titration calorimetric analysis | Homo sapiens | 1 | ALA3769341 | assay format | Scientific Literature | |
| 12. | ALA3772744 | B | Binding affinity to recombinant His6-TEV fused human BAZ2A assessed as melting temperature shift at 10 uM by real time PCR analysis | Homo sapiens | 1 | ALA3769341 | single protein format | Scientific Literature | |
| 13. | ALA3773108 | B | Binding affinity to biotinylated C-terminal Avi/His-TEV-tagged BAZ2A (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
| 14. | ALA3773290 | B | Binding affinity to BAZ2A in human HUT78 cell extract by chemoproteomic competition binding assay | Homo sapiens | 1 | ALA3769341 | cell-based format | Scientific Literature | |
| 15. | ALA3773292 | B | Binding affinity to BAZ2A in human HUT78 cell extract up to 50 uM by chemoproteomic competition binding assay | Homo sapiens | 1 | ALA3769341 | cell-based format | Scientific Literature | |
| 16. | ALA3773296 | B | Binding affinity to N-terminal eGFP tagged BAZ2A (unknown origin) expressed in HDAC inhibitor SAHA-treated human U2OS cells assessed as acceleration of FRAP half-recovery time at 1 uM incubated for 24 hrs | Homo sapiens | 2 | ALA3769341 | cell-based format | Scientific Literature | |
| 17. | ALA3773297 | B | Binding affinity to N-terminal eGFP tagged BAZ2A N1873F mutant (unknown origin) expressed in HDAC inhibitor SAHA-treated human U2OS cells assessed as acceleration of FRAP half-recovery time at 1 uM incubated for 24 hrs | Homo sapiens | 1 | ALA3769341 | cell-based format | Scientific Literature | |
| 18. | ALA3779311 | B | Inhibition of recombinant human BAZ2A expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 19. | ALA4020272 | B | Binding affinity to human BAZ2A (M1792 to L1905 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 1 | ALA4017535 | assay format | Scientific Literature | |
| 20. | ALA4038414 | B | Inhibition of human BAZ2A (M1792 to L1905 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 3 | ALA4038268 | assay format | Scientific Literature |
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