| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3111500 | B | Binding affinity to BRPF3 bromodomain (unknown origin) assessed as change in melting temperature at 10 uM by differential scanning fluorimetric analysis | Homo sapiens | 35 | ALA3108763 | single protein format | Scientific Literature | |
| 2. | ALA3134634 | B | Binding affinity to BRPF3 (unknown origin) at 4 uM by thermal shift assay | Homo sapiens | 3 | ALA3132771 | single protein format | Scientific Literature | |
| 3. | ALA3385107 | B | Binding affinity to 6H-Flag-tagged Tev-BRPF3 (579-706 aa) (unknown origin) by TR-FRET competitive assay | Homo sapiens | 1 | ALA3352488 | single protein format | Scientific Literature | |
| 4. | ALA3383421 | B | Inhibition of human BRPF3 by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
| 5. | ALA3591381 | B | Binding affinity to BRPF3 (unknown origin) by BROMOscan panel based assay | Homo sapiens | 1 | ALA3588744 | single protein format | Scientific Literature | |
| 6. | ALA3757235 | B | Binding affinity to BRPF3 (unknown origin) by isothermal titration calorimetry | Homo sapiens | 1 | ALA3751772 | single protein format | Scientific Literature | |
| 7. | ALA3771494 | B | Inhibition of BRPF3 (unknown origin) by Alpha Screen assay | Homo sapiens | 1 | ALA3769336 | single protein format | Scientific Literature | |
| 8. | ALA3779323 | B | Binding affinity to recombinant human BRPF3 expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 9. | ALA3790875 | B | Binding affinity to BRPF3 (unknown origin) by isothermal titration calorimetric analysis | Homo sapiens | 2 | ALA3785033 | single protein format | Scientific Literature | |
| 10. | ALA3830586 | B | Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6HisFlag-Tev-BRPF3 (579 to 706 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells after 30 mins by TR-FRET assay | Homo sapiens | 1 | ALA3826893 | cell-based format | Scientific Literature | |
| 11. | ALA4003560 | B | Binding affinity to human partial length BRPF3 expressed in bacterial expression system by BROMOscan method | Homo sapiens | 1 | ALA4002593 | assay format | Scientific Literature | |
| 12. | ALA4020275 | B | Binding affinity to human BRPF3 (E588 to G701 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 1 | ALA4017535 | assay format | Scientific Literature | |
| 13. | ALA4030909 | B | Inhibition of human BRPF3 (588 to 701 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assay | Homo sapiens | 16 | ALA4028852 | assay format | Scientific Literature | |
| 14. | ALA4030917 | B | Inhibition of His-tagged BRPF3 (unknown origin) using [H-YSGRGKacGGKacGLGKacGGAKacRHRK(Biotin)-OH peptide as substrate by alphaScreen assay | Homo sapiens | 1 | ALA4028852 | single protein format | Scientific Literature | |
| 15. | ALA4030945 | B | Binding affinity to BRPF3 (unknown origin) by isothermal titration calorimetry | Homo sapiens | 1 | ALA4028852 | single protein format | Scientific Literature | |
| 16. | ALA4038417 | B | Inhibition of human BRPF3 (E588 to G701 residues) expressed in bacterial expression system by BROMOscan assay | Homo sapiens | 3 | ALA4038268 | assay format | Scientific Literature | |
| 17. | ALA4047545 | B | Inhibition of human partial length BRPF3 (E588 to G701 residues) expressed in bacterial expression system assessed as residual activity at 500 nM relative to control by BROMOscan assay | Homo sapiens | 1 | ALA4043246 | assay format | Scientific Literature | |
| 18. | ALA4051533 | B | Inhibition of BRPF3 (592 to 711 residues) (unknown origin) preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,12 diacetylated histone H4 (1 to 20 residues) peptide as substrate measured after 1 hr by TR-FRET assay | Homo sapiens | 3 | ALA4049437 | single protein format | Scientific Literature | |
| 19. | ALA4051561 | B | Inhibition of BRPF3 (592 to 711 residues) (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO Orange-dye based fluorescence thermal shift assay | Homo sapiens | 1 | ALA4049437 | single protein format | Scientific Literature | |
| 20. | ALA4051605 | B | Inhibition of BRPF3 (592 to 711 residues) (unknown origin) using biotin-acetylated histone H4 peptide as substrate after 30 mins by AlphaScreen assay | Homo sapiens | 2 | ALA4049437 | single protein format | Scientific Literature |
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