# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2209120 | B | Inhibition of PRC2 complex of EZH1, EED, SUZ12, AEBP2 and RbAp48 using histone H3 peptide (21 to 44) as substrate and [3H]SAM after 1 hr by SPA | 3 | ALA2202955 | protein complex format | Scientific Literature | ||
2. | ALA3111735 | B | Inhibition of EZH1/EED/SUZ12/AEBP2/RBBP4 complex (unknown origin)-mediated incorporation of methyl group from [3H]-SAM into peptide substrate up to 50 uM by scintillation proximity assay | Homo sapiens | 1 | ALA3108684 | protein complex format | Scientific Literature | |
3. | ALA4144878 | B | Inhibition of human N-terminal His-tagged EZH2/flag-tagged EED/SUZ12/AEBP2/RBAP48 A677G mutant (2 to end residues) expressed in baculovirus infected Sf9 insect cells using histone H3 (1 to 50 residues)-GGK as substrate after 2 hrs in presence of SAM by fluorescence assay | Homo sapiens | 25 | ALA4138300 | cell-based format | Scientific Literature |