| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3226588 | B | Binding affinity to TAF1 bromodomain-2 (unknown origin) assessed as change in melting temperature at 10 uM by differential scanning fluorimetric analysis | Homo sapiens | 1 | ALA3217564 | single protein format | Scientific Literature | |
| 2. | ALA3267587 | B | Binding affinity to TAF1(2) (unknown origin) by thermal shift assay | Homo sapiens | 2 | ALA3259646 | single protein format | Scientific Literature | |
| 3. | ALA3383430 | B | Inhibition of human TAF1 by BROMOscan assay | Homo sapiens | 1 | ALA3351476 | single protein format | Scientific Literature | |
| 4. | ALA3380072 | B | Binding affinity to TAF1 (unknown origin) by bromodomain displacement assay | Homo sapiens | 1 | ALA3351605 | single protein format | Scientific Literature | |
| 5. | ALA3583523 | B | Binding affinity to biotinylated TAF1B2 (155 to 276 amino acid residues) (unknown origin) expressed in Rosetta2 cells by bio-layer interferometry method | Homo sapiens | 1 | ALA3580597 | cell-based format | Scientific Literature | |
| 6. | ALA3591377 | B | Binding affinity to TAF1 (unknown origin) by BROMOscan panel based assay | Homo sapiens | 1 | ALA3588744 | single protein format | Scientific Literature | |
| 7. | ALA3591401 | B | Binding affinity to TAF1 in human HUT78 cells incubated for 45 mins by mass spectrometry based bromosphere chemoproteomic assay | Homo sapiens | 3 | ALA3588744 | cell-based format | Scientific Literature | |
| 8. | ALA3773281 | B | Binding affinity to biotinylated TAF1 bromodomain-1 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
| 9. | ALA3773282 | B | Binding affinity to biotinylated TAF1 bromodomain-2 (unknown origin) expressed in Escherichia coli at 0.2 to 1 uM by Biolayer Interferometric analysis | Homo sapiens | 2 | ALA3769341 | assay format | Scientific Literature | |
| 10. | ALA3779325 | B | Binding affinity to recombinant human TAF1 bromodomain 2 expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 11. | ALA3782789 | B | Binding affinity to human His6-tagged TAF1 bromodomain 1 (R1377 to D1503 residues) expressed in Escherichia coli BL21(DE3) cells at 200 uM incubated for 30 mins by SYPRO orange staining based fluorescence thermal shift assay | Homo sapiens | 16 | ALA3779865 | cell-based format | Scientific Literature | |
| 12. | ALA3821664 | B | Binding affinity to human TAF1 expressed in Escherichia coli BL21(DE3)-R3-pRARE2 assessed as change in melting temperature at 25 uM by SYPRO orange based protein stability shift assay | Homo sapiens | 10 | ALA3817837 | assay format | Scientific Literature | |
| 13. | ALA3863020 | B | Binding affinity to TAF1 bromodomain 1 (unknown origin) assessed as change in melting temperature at 100 uM by differential scanning fluorimetric assay | Homo sapiens | 1 | ALA3861991 | single protein format | Scientific Literature | |
| 14. | ALA3863021 | B | Binding affinity to TAF1 bromodomain 2 (unknown origin) assessed as change in melting temperature at 100 uM by differential scanning fluorimetric assay | Homo sapiens | 1 | ALA3861991 | single protein format | Scientific Literature | |
| 15. | ALA3864415 | B | Displacement of biotinylated ligand from recombinant His-tagged TAF1 bromodomain 1 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 2 | ALA3864133 | single protein format | Scientific Literature | |
| 16. | ALA3864416 | B | Displacement of biotinylated ligand from recombinant His-tagged TAF1 bromodomain 2 (unknown origin) measured after 10 mins by TR-FRET assay | Homo sapiens | 2 | ALA3864133 | single protein format | Scientific Literature | |
| 17. | ALA4047556 | B | Inhibition of human partial length TAF1 BD2 (D1521 to D1656 residues) expressed in bacterial expression system assessed as residual activity at 500 nM relative to control by BROMOscan assay | Homo sapiens | 1 | ALA4043246 | assay format | Scientific Literature | |
| 18. | ALA4051534 | B | Inhibition of human GST-tagged TAF1 BD2 (1519 to 1651 residues) expressed in Escherichia coli BL21 (DE3)-R3-pRARE2 preincubated for 15 mins followed by addition of C-terminal biotinylated synthetic K5,8,12,16 tetra-acetylated histone H4 (1 to 20 residues) peptide as substrate measured after 1 hr by TR-FRET assay | Homo sapiens | 24 | ALA4049437 | assay format | Scientific Literature | |
| 19. | ALA4051582 | B | Inhibition of TAF1 BD2 (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO Orange-dye based fluorescence thermal shift assay | Homo sapiens | 1 | ALA4049437 | single protein format | Scientific Literature | |
| 20. | ALA4051583 | B | Inhibition of TAF1 BD1 (unknown origin) assessed as change in melting temperature at 10 uM by SYPRO Orange-dye based fluorescence thermal shift assay | Homo sapiens | 1 | ALA4049437 | single protein format | Scientific Literature |
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