| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2339960 | B | Inhibition of Kallikrein-14 (unknown origin) using VPR-AMC substrate incubated for 15 mins prior to substrate addition measured for 2 hrs | Homo sapiens | 1 | ALA2331221 | single protein format | Scientific Literature | |
| 2. | ALA2339090 | B | Inhibition of Kallikrein-14 (unknown origin) using VPR-AMC substrate assessed as residual activity at 10 uM incubated for 15 mins prior to substrate addition measured for 2 hrs | Homo sapiens | 1 | ALA2331221 | single protein format | Scientific Literature | |
| 3. | ALA2412635 | B | Binding affinity to human kallikrein 14 assessed as half life of deacylated enzyme | Homo sapiens | 3 | ALA2406906 | single protein format | Scientific Literature | |
| 4. | ALA2412648 | B | Inhibition of human kallikrein 14 measured after 15 mins at pH 8 by fluorescence assay | Homo sapiens | 7 | ALA2406906 | single protein format | Scientific Literature | |
| 5. | ALA3100873 | B | Reversible inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 to 60 mins by fluorescence assay | Homo sapiens | 16 | ALA3098059 | single protein format | Scientific Literature | |
| 6. | ALA3100878 | B | Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate at 50 uM after 15 mins by fluorescence assay | Homo sapiens | 8 | ALA3098059 | single protein format | Scientific Literature | |
| 7. | ALA3100879 | B | Inhibition of human kallikrein14 using Boc-Val-Pro-Arg-AMC as substrate after 15 mins by fluorescence assay | Homo sapiens | 8 | ALA3098059 | single protein format | Scientific Literature | |
| 8. | ALA3413943 | B | Inhibition of human KLK14 using Boc-Val-Pro-Arg-AMC as substrate at 50 uM after 15 mins by fluorescence assay | Homo sapiens | 2 | ALA3407351 | single protein format | Scientific Literature | |
| 9. | ALA3626834 | B | Inhibition of KLK14 (unknown origin) expressed in Sf9 cells at 25 nM using Ac-YANR-pNA substrate by spectrophotometry method | Homo sapiens | 7 | ALA3621201 | cell-based format | Scientific Literature | |
| 10. | ALA3627278 | B | Inhibition of KLK14 (unknown origin) expressed in Sf9 cells using Ac-YANR-pNA substrate by spectrophotometry method | Homo sapiens | 4 | ALA3621201 | cell-based format | Scientific Literature | |
| 11. | ALA4038144 | B | Inhibition of recombinant human C-terminal 10His-tagged KLK14 (19 to 248 residues) expressed in mouse NS0 cells using fluorogenic Boc-VPR-AMC peptide as substrate by fluorescence based assay | Homo sapiens | 3 | ALA4033799 | cell-based format | Scientific Literature | |
| 12. | ALA4201847 | B | Inhibition of KLK14 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured after 30 mins by fluorescence based assay | Homo sapiens | 2 | ALA4196210 | assay format | Scientific Literature | |
| 13. | ALA4330020 | B | Inhibition of KLK14 (unknown origin) expressed in sf9 cells using Ac-YANR-pNA as substrate preincubated for 30 mins followed by substrate addition and measured for 7 mins by spectrophotometric method | Homo sapiens | 3 | ALA4325933 | cell-based format | Scientific Literature | |
| 14. | ALA4355185 | B | Inhibition of recombinant human KLK14 expressed in Spodoptera frugiperda Sf9 cells using Boc-QAR-MCA as susbtrate measured every 60 secs for 10 mins by fluorescence based assay | Homo sapiens | 3 | ALA4354795 | cell-based format | Scientific Literature | |
| 15. | ALA4355189 | B | Inhibition of recombinant KLK14 (unknown origin) expressed in Spodoptera frugiperda Sf9 cells using pNA peptide as susbtrate measured every 10 secs for 300 secs by spectrophotometric analysis | Homo sapiens | 1 | ALA4354795 | cell-based format | Scientific Literature | |
| 16. | ALA4388468 | A | Inhibition of recombinant C-terminal 10His-tagged human KLK14 (Gln19 to Met248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate after 40 mins by fluorescence intensity assay | Homo sapiens | 1 | ALA4387717 | cell-based format | Scientific Literature | |
| 17. | ALA4400466 | B | Inhibition of recombinant human C-terminal 10-His-tagged KLK14 (Q19 to M248 residues) expressed in mouse NS0 cells using BOC-VPR-AMC as substrate incubated for 40 mins by FLINT assay | Homo sapiens | 15 | ALA4396973 | cell-based format | Scientific Literature | |
| 18. | ALA4424184 | B | Inhibition of KLK14 (unknown origin) at 100 uM using Boc-Val-Pro-Arg- AMC substrate incubated for 15 mins by fluorescence assay | Homo sapiens | 1 | ALA4422656 | single protein format | Scientific Literature | |
| 19. | ALA4424187 | B | Inhibition of recombinant human KLK14 using S-2302 substrate | Homo sapiens | 1 | ALA4422656 | single protein format | Scientific Literature | |
| 20. | ALA4831733 | B | Inhibition of KLK14 (unknown origin) assessed as inhibition of release of AMC fluorescent product using H-VPR-AMC as substrate at 10 uM incubated for 30 mins by microplate reader relative to control | Homo sapiens | 7 | ALA4831480 | single protein format | Scientific Literature |
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