#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA765806	B	Inhibitory activity against purified fusion of maltose binding with PHD1 as enzyme and (HIF) human prolyl hydroxylases as substrate		1		single protein format	Scientific Literature
2.	ALA2045987	B	Inhibition of PHD1		56		single protein format	Scientific Literature
3.	ALA1942541	B	Inhibition of PHD1		3		single protein format	Scientific Literature
4.	ALA946278	B	Inhibition of human recombinant HIF PHD1	Homo sapiens	2		single protein format	Scientific Literature
5.	ALA1219076	B	Inhibition of human recombinant PHD1 expressed in Sf9 cells by time-resolved fluorescence assay	Homo sapiens	15		cell-based format	Scientific Literature
6.	ALA1243624	B	Activity of HIF prolyl hydroxylase-1		3		single protein format	Scientific Literature
7.	ALA1260833	B	Inhibition of PHD1 by HTRF assay		8		single protein format	Scientific Literature
8.	ALA3118614	B	Inhibition of PHD1 (unknown origin) expressed in Sf9 cells using HIF-1alpha peptide as substrate preincubated for 30 mins followed by substrate addition measured after 2 hrs by HTRF assay in presence of 2-oxoglutarate	Homo sapiens	1		cell-based format	Scientific Literature
9.	ALA3705564	B	Inhibition Assay: Hydroxylated HIF bonds specifically to the von Hippel-Lindau protein-elongin B-elongin C complex (VBC complex). This interaction occurs only if HIF is hydroxylated on a conserved prolyl radical. It is the basis for the biochemical determination of HIF prolyl hydroxylase activity. The test is carried out as described [Oehme F., Jonghaus W., Narouz-Ott L., Huetter J., Flamme I., Anal. Biochem. 330 (1), 74-80 (2004)].	Homo sapiens	20		single protein format	BindingDB Database
10.	ALA3862231	B	Inhibition of recombinant human HIF-PHD1 expressed in insect Sf9 cells using biotinyl-DLDLEMLAPYIPMDDDFQL as substrate after 60 mins by DELFIA	Homo sapiens	1		cell-based format	Scientific Literature
11.	ALA3888867	B	HIF-PH Assay: Ketoglutaric acid α-[1-14C]-sodium salt, alpha-ketoglutaric acid sodium salt, and HPLC purified peptide may be obtained from commercial sources, e.g., Perkin-Elmer (Wellesley Mass.), Sigma-Aldrich, and SynPep Corp. (Dublin Calif.), respectively. Peptides for use in the assay may be fragments of HIFα as described above or as disclosed in International Publication WO 2005/118836, incorporated by reference herein. HIF-pH, e.g., PHD1 (EGLN2) or PHD2 (EGLN1), can be expressed in, e.g., insect Hi5 cells, and partially purified, e.g., through a SP ion exchange chromatography column. Enzyme activity is determined by capturing 14CO2 using an assay described by Kivirikko and Myllyla (1982, Methods Enzymol. 82:245-304). Assay reactions contain 50 mM HEPES (pH 7.4), 100 μM α-ketoglutaric acid sodium salt, 0.30 mCi/mL ketoglutaric acid α-[1-14C]-sodium salt, 40 μM FeSO4, 1 mM ascorbate, 1541.8 units/mL Catalase, with or without 50 μM peptide substrate and various concentrations of compound of the invention. Reactions are initiated by addition of HIF-PH enzyme.	Homo sapiens	183		cell-based format	BindingDB Database
12.	ALA4017304	B	Inhibition of full length HIF-PHD1 (unknown origin) expressed in baculovirus infected sf9 cells using DLDLEMLAPYIPMDDDFQL/2-Oxoglutarate as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins by UPLC-MS analysis	Homo sapiens	66		cell-based format	Scientific Literature
13.	ALA4149385	B	Inhibition of HIF-PHD1 (unknown origin) expressed in insect Hi5 cells using peptide as substrate	Homo sapiens	1		cell-based format	Scientific Literature
14.	ALA4149396	B	Inhibition of PHD1 (unknown origin)	Homo sapiens	1		single protein format	Scientific Literature
15.	ALA4149404	B	Inhibition of FLAG- tagged full length HIF-PHD1 (unknown origin) expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL as substrate preincubated for 30 mins followed by substrate addition measured after 2 hrs by LANCE assay	Homo sapiens	1		cell-based format	Scientific Literature
16.	ALA4149411	B	Inhibition of recombinant human HIF-PHD1 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL as substrate preincubated for 60 mins followed by substrate addition measured after 60 mins by TR-FRET assay	Homo sapiens	1		cell-based format	Scientific Literature
17.	ALA4329853	B	Inhibition of recombinant human HIF-PHD1 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL and 2-oxoglutarate as substrates preincubated for 30 mins followed by substrates addition and measured after 2 hrs by TR-FRET assay	Homo sapiens	27		cell-based format	Scientific Literature
18.	ALA4766453	B	Inhibition of FLAG-tagged full-length HIF-PHD1 (unknown origin) expressed in baculovirus infected Sf9 cells using 2-oxoglutarate and HIF1alpha biotinyl-DLDLEMLAPYIPMDDDFQL as peptide substrates preincubated for 30 mins followed by substrate addition and measured after 2 hrs by LANCE assay	Homo sapiens	1		cell-based format	Scientific Literature
19.	ALA4831469	B	Inhibition of recombinant full length human N-terminal FLAG-tagged PHD1 expressed in baculovirus expression system using HIF1/C35 complex as substrate preincubated for 30 mins followed by substrate addition measured after 10 mins by TR-FRET assay	Homo sapiens	6		assay format	Scientific Literature
20.	ALA5229126	B	Inhibition of human PHD1 expressed in H5 insect cells	Homo sapiens	5		cell-based format	Scientific Literature