# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA704110 | B | Inhibition of Janus kinase 1 | 1 | ALA1136271 | single protein format | Scientific Literature | ||
2. | ALA857179 | B | Inhibition of Janus kinase 1 | 2 | ALA1133428 | single protein format | Scientific Literature | ||
3. | ALA860904 | B | Average Binding Constant for JAK1 (Kin.Dom. 1); NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
4. | ALA910181 | B | Inhibition of Jak1 | Homo sapiens | 1 | ALA1141381 | single protein format | Scientific Literature | |
5. | ALA1019239 | B | Inhibition of IFN-alpha-induced JAK1 Y1022/1023 phosphorylation in serum starved human U266 cells by Western blot analysis | Homo sapiens | 1 | ALA1155075 | cell-based format | Scientific Literature | |
6. | ALA1020094 | B | Inhibition of JAK1 at 1 uM | 1 | ALA1155075 | single protein format | Scientific Literature | ||
7. | ALA1020097 | B | Inhibition of JAK1 at 10 uM | 1 | ALA1155075 | single protein format | Scientific Literature | ||
8. | ALA990527 | B | Inhibition of Jak1 | 1 | ALA1149823 | single protein format | Scientific Literature | ||
9. | ALA987115 | B | Inhibition of JAK1 | 1 | ALA1142524 | single protein format | Scientific Literature | ||
10. | ALA1025742 | B | Binding affinity to human JAK1 at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
11. | ALA1016954 | B | Inhibition of JAK1 | 4 | ALA1152817 | single protein format | Scientific Literature | ||
12. | ALA1019776 | B | Inhibition of JAK1 | 1 | ALA1151738 | single protein format | Scientific Literature | ||
13. | ALA1054874 | B | Inhibition of JAK1 at 10 uM by HotSpot assay relative to control | 1 | ALA1153464 | single protein format | Scientific Literature | ||
14. | ALA1057717 | B | Binding constant for JAK1(Kin.Dom.1/JH2 - pseudokinase) kinase domain | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
15. | ALA1053757 | B | Inhibition of JAK1 kinase domain 1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
16. | ALA1053758 | B | Inhibition of JAK1 kinase domain 2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
17. | ALA1040927 | B | Inhibition of human recombinant JAK1 | Homo sapiens | 1 | ALA1156112 | single protein format | Scientific Literature | |
18. | ALA1038360 | B | Inhibition of Jak1 | 1 | ALA1155349 | single protein format | Scientific Literature | ||
19. | ALA1072206 | B | Inhibition of JAK1 | 3 | ALA1157561 | single protein format | Scientific Literature | ||
20. | ALA1102771 | B | Inhibition of GST-tagged JAK1 assessed as inhibition of biotinylated IRS1 substrate phosphorylation after 60 mins by caliper mobility shift assay | 16 | ALA1154949 | single protein format | Scientific Literature |