| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA704110 | B | Inhibition of Janus kinase 1 | 1 | single protein format | Scientific Literature | |||
| 2. | ALA857179 | B | Inhibition of Janus kinase 1 | 2 | single protein format | Scientific Literature | |||
| 3. | ALA860904 | B | Average Binding Constant for JAK1 (Kin.Dom. 1); NA=Not Active at 10 uM | Homo sapiens | 20 | single protein format | Scientific Literature | ||
| 4. | ALA910181 | B | Inhibition of Jak1 | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA1815193 | B | Inhibition of JAK1 phosphorylation in human A2780 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA1799027 | B | Inhibition of JAK1 at 10 uM | 2 | single protein format | Scientific Literature | |||
| 7. | ALA2014442 | B | Inhibition of JAK1 at 10 uM | 1 | single protein format | Scientific Literature | |||
| 8. | ALA2019648 | B | Inhibition of JAK1 assessed as remaining activity at 0.1 uM by radiolabeled kinase assay relative to control | 1 | single protein format | Scientific Literature | |||
| 9. | ALA1827269 | B | Activity of JAK1 JH2 pseudokinase domain kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
| 10. | ALA1828387 | B | Activity of JAK1 JH1 catalytic domain kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
| 11. | ALA2033415 | B | Inhibition of JAK1 in human HEK293 cells after 1 hr by competition binding assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA2032472 | B | Inhibition of JAK1 | 2 | single protein format | Scientific Literature | |||
| 13. | ALA2039968 | B | Inhibition of recombinant JAK1 using poly(Glu,Ala,Tyr) as substrate after 2 hrs by luminometric assay | 22 | single protein format | Scientific Literature | |||
| 14. | ALA2067180 | B | Inhibition of human JAK1 expressed in baculovirus using biotinyl-amino-hexanoyl-EQEDEPEGDYFEWLE-amide as substrate preincubated for 1 hr measured after 20 mins by time resolved fluorescence assay | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 15. | ALA1962116 | B | GSK_PKIS: JAK1 mean inhibition at 0.1 uM [Nanosyn] | 366 | single protein format | GSK Published Kinase Inhibitor Set | |||
| 16. | ALA1962117 | B | GSK_PKIS: JAK1 mean inhibition at 1 uM [Nanosyn] | 366 | single protein format | GSK Published Kinase Inhibitor Set | |||
| 17. | ALA1785329 | B | Inhibition of human JAK1 using poly[Glu:Tyr] by Hotspot assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA1787836 | B | Inhibition of JAK1 at 10 uM | 1 | single protein format | Scientific Literature | |||
| 19. | ALA1019239 | B | Inhibition of IFN-alpha-induced JAK1 Y1022/1023 phosphorylation in serum starved human U266 cells by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA1020094 | B | Inhibition of JAK1 at 1 uM | 1 | single protein format | Scientific Literature |
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