# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA1019784 | B | Binding affinity to RPS6KA6 kinase domain.2- C-terminal | 1 | single protein format | Scientific Literature | |||
2. | ALA1039275 | B | Binding constant for RPS6KA6(Kin.Dom.1 - C-terminal) kinase domain | Homo sapiens | 38 | single protein format | Scientific Literature | ||
3. | ALA1061926 | B | Binding constant for RPS6KA6(Kin.Dom.2 - N-terminal) kinase domain | Homo sapiens | 38 | single protein format | Scientific Literature | ||
4. | ALA1043888 | B | Binding affinity to RSK4 kinase domain 2 C-terminal assessed as percentage of kinase remaining bound to the bead at 1 uM by T7 phage display based binding assay | 1 | single protein format | Scientific Literature | |||
5. | ALA1052961 | B | Inhibition of RPS6KA6 kinase domain 1 assessed as enzyme activity at 1 uM relative to untreated control | 1 | single protein format | Scientific Literature | |||
6. | ALA1052962 | B | Inhibition of RPS6KA6 kinase domain 2 assessed as enzyme activity at 1 uM relative to untreated control | 1 | single protein format | Scientific Literature | |||
7. | ALA1036948 | B | Inhibition of RSK4 at 1 uM | 1 | single protein format | Scientific Literature | |||
8. | ALA1043807 | B | Residual activity of RPS6KA6 at 1 uM by microplate scintillation counting | 3 | single protein format | Scientific Literature | |||
9. | ALA1072514 | B | Residual activity of RPS6KA6 at 0.1 uM by microplate scintillation counting | 3 | single protein format | Scientific Literature | |||
10. | ALA1071367 | B | Residual activity of RPS6KA6 at 10 uM by microplate scintillation counting | 3 | single protein format | Scientific Literature | |||
11. | ALA1101761 | B | Inhibition of RSK4 at 10 uM | 2 | single protein format | Scientific Literature | |||
12. | ALA1103235 | B | Inhibition of RSK4 at 5 uM | 1 | single protein format | Scientific Literature | |||
13. | ALA1167695 | B | Inhibition of RPS6KA6 N-terminal domain1 at 1 uM | 10 | single protein format | Scientific Literature | |||
14. | ALA1167696 | B | Inhibition of RPS6KA6 C-terminal domain2 at 1 uM | 10 | single protein format | Scientific Literature | |||
15. | ALA1175331 | B | Inhibition of RSK4 N-terminal domain1 at 10 uM | 2 | single protein format | Scientific Literature | |||
16. | ALA1175332 | B | Inhibition of RSK4 C-terminal domain2 at 10 uM | 2 | single protein format | Scientific Literature | |||
17. | ALA1244286 | B | Inhibition of RSK4 at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 5 | single protein format | Scientific Literature | |||
18. | ALA1244973 | B | Binding affinity to RPS6KA6(Kin.Dom.1-N-terminal) | 7 | single protein format | Scientific Literature | |||
19. | ALA1244974 | B | Binding affinity to RPS6KA6(Kin.Dom.2-C-terminal) | 7 | single protein format | Scientific Literature | |||
20. | ALA1251686 | B | Inhibition of RPS6KA6 at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | single protein format | Scientific Literature |