# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3361954 | B | Agonist activity at human TAS2R16 expressed in U2OS cells by summary (Abse5) assay | Homo sapiens | 1 | ALA3351646 | cell-based format | Scientific Literature | |
2. | ALA3361955 | B | Antagonist activity at human TAS2R16 expressed in U2OS cells by Ga16gust44 Clone 7A FLIPR/summary (Abse5) assay | Homo sapiens | 1 | ALA3351646 | cell-based format | Scientific Literature | |
3. | ALA4346431 | F | Antagonist activity at recombinant human TAS2R16 transiently expressed in HEK293T co-expressing Galpha16gust44 assessed as inhibition of salicin-induced intracellular calcium level by measuring remaining activity at 25 uM by fluo-4AM dye based FLIPR assay relative to control | Homo sapiens | 2 | ALA4342523 | cell-based format | Scientific Literature | |
4. | ALA4417701 | F | Antagonist activity at full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 25 uM in presence of 10 mM phenyl-beta-glucopyranoside by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
5. | ALA4417702 | F | Antagonist activity at full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 25 uM in presence of 5 mM phenyl-beta-glucopyranoside by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
6. | ALA4417703 | F | Antagonist activity at full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 25 uM in presence of 2.5 mM phenyl-beta-glucopyranoside by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
7. | ALA4417704 | F | Antagonist activity at full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 25 uM in presence of 1.25 mM phenyl-beta-glucopyranoside by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
8. | ALA4417705 | F | Antagonist activity at full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 25 uM in presence of 0.625 mM phenyl-beta-glucopyranoside by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
9. | ALA4417706 | F | Antagonist activity at full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 25 uM in presence of 0.3125 mM phenyl-beta-glucopyranoside by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
10. | ALA4417707 | F | Antagonist activity at full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 25 uM in presence of 0.1563 mM phenyl-beta-glucopyranoside by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
11. | ALA4417708 | F | Antagonist activity at full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 25 uM in presence of 0.0781 mM phenyl-beta-glucopyranoside by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
12. | ALA4417709 | F | Antagonist activity at full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 25 uM in presence of 0.0391 mM phenyl-beta-glucopyranoside by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
13. | ALA4417710 | F | Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 10 mM by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
14. | ALA4417711 | F | Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 5 mM by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
15. | ALA4417712 | F | Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 2.5 mM by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
16. | ALA4417713 | F | Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 1.25 mM by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
17. | ALA4417714 | F | Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 0.625 mM by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
18. | ALA4417715 | F | Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 0.3125 mM by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
19. | ALA4417716 | F | Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 0.1563 mM by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data | |
20. | ALA4417717 | F | Activation of full-length human TAS2R16 expressed in HEK293T/Galpha16-gustducin 44 cells assessed as effect on calcium flux by measuring deltaF/F0 ratio at 0.0781 mM by Fluo-4 dye based FLIPR assay | Homo sapiens | 1 | ALA4417621 | cell-based format | Patent Bioactivity Data |