| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3361957 | B | Agonist activity at human TAS2R41 expressed in U2OS cells by Ga16gust44 Clone 7A FLIPR/summary (Abse5) assay | Homo sapiens | 1 | ALA3351646 | cell-based format | Scientific Literature | |
| 2. | ALA4346435 | F | Antagonist activity at recombinant human TAS2R41 transiently expressed in HEK293T co-expressing Galpha16gust44 assessed as inhibition of picric acid-induced intracellular calcium level by measuring remaining activity at 25 uM by fluo-4AM dye based FLIPR assay relative to control | Homo sapiens | 2 | ALA4342523 | cell-based format | Scientific Literature | |
| 3. | ALA4419016 | F | Agonist activity at recombinant human N-terminal rat ST3 receptor-fused TAS2R41 expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level at 100 uM by FLIPR assay | Homo sapiens | 1 | ALA4418912 | cell-based format | Patent Bioactivity Data | |
| 4. | ALA4419220 | F | Agonist activity at human TAS2R41 expressed in HEK293T cells co-expressing Galpha15 assessed as increase in intracellular calcium level by Calcium-3 dye based fluorescence assay | Homo sapiens | 1 | ALA4419163 | cell-based format | Patent Bioactivity Data | |
| 5. | ALA4419245 | F | Agonist activity at human TAS2R41 expressed in HEK293T cells co-expressing Galpha15 assessed as increase in intracellular calcium level at 20 mM by Calcium-3 dye based fluorescence assay relative to control | Homo sapiens | 3 | ALA4419163 | cell-based format | Patent Bioactivity Data | |
| 6. | ALA4421753 | F | Agonist activity at recombinant human N-terminal rat ST3 receptor-fused TAS2R41 expressed in HEK293T cells co-expressing Galpha16gust44 assessed as effect on intracellular calcium level at 100 uM by FLIPR assay | Homo sapiens | 1 | ALA4421717 | cell-based format | Patent Bioactivity Data | |
| 7. | ALA4482402 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 80 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.146471 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 8. | ALA4482403 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 75 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.132941 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 9. | ALA4482404 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 70 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.152941 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 10. | ALA4482405 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 65 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.138235 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 11. | ALA4482406 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 60 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.145294 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 12. | ALA4482407 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 55 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.168235 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 13. | ALA4482408 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 50 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.167647 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 14. | ALA4482409 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 45 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.176471 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 15. | ALA4482410 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 40 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.171765 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 16. | ALA4482411 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 35 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.167647 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 17. | ALA4482412 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 30 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.166471 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 18. | ALA4482413 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-5) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 25 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.158824 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 19. | ALA4482414 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-7) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 80 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.146471 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data | |
| 20. | ALA4482415 | F | Agonist activity at N-terminal rat ST3 receptor-fused full length human TAS2R41 (nucleotide sequence ID No-7) expressed in HEK293T cells co-expressing Galpha16gust44 assessed as increase in intracellular calcium level by measuring deltaF/F0 ratio level at 75 mM by Fluo-4AM dye based FLIPR assay (Rvb = 0.132941 No_unit) | Homo sapiens | 1 | ALA4482304 | cell-based format | Patent Bioactivity Data |
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