| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3371276 | B | Inhibition of proteasome subunit beta-2i in human Raji cells using BODIPY- epoxomicin by fluorescent densitometry | Homo sapiens | 13 | ALA3351747 | cell-based format | Scientific Literature | |
| 2. | ALA3371285 | B | Inhibition of proteasome subunit beta-2i in human RPMI8226 cells using BODIPY-epoxomicin by fluorescent densitometry | Homo sapiens | 8 | ALA3351747 | cell-based format | Scientific Literature | |
| 3. | ALA3997514 | B | Inhibition of MECL1 in human MOLT4 cell lysate after 1 hr by ELISA | Homo sapiens | 4 | ALA3994666 | assay format | Scientific Literature | |
| 4. | ALA4123724 | B | Inhibition of human 20S immunoproteasome beta-2 using Bz-VGR-AMC as substrate after 60 mins by fluorescence assay | Homo sapiens | 9 | ALA4118199 | single protein format | Scientific Literature | |
| 5. | ALA4255072 | B | Inhibition of human 20S immunoproteasome beta-2 using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assay | Homo sapiens | 16 | ALA4251654 | single protein format | Scientific Literature | |
| 6. | ALA4255074 | B | Inhibition of human 20S immunoproteasome beta-2 at 50 uM using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assay relative to control | Homo sapiens | 31 | ALA4251654 | single protein format | Scientific Literature | |
| 7. | ALA4255079 | B | Activation of human 20S immunoproteasome beta-2 at 50 uM using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assay relative to control | Homo sapiens | 4 | ALA4251654 | single protein format | Scientific Literature | |
| 8. | ALA4310879 | B | Inhibition of 20s immunoproteasome MECL1 in human erythrocytes using Suc-Leu-Leu-ValTyr-MCA as substrate preincubated for 10 mins followed by substrate addition and measured after 6 hrs by fluorescence assay | Homo sapiens | 1 | ALA4308881 | cell-based format | Scientific Literature | |
| 9. | ALA4310881 | B | Inhibition of 20s immunoproteasome MECL1 in human erythrocytes at 15 uM using Suc-Leu-Leu-ValTyr-MCA as substrate preincubated for 10 mins followed by substrate addition and measured after 6 hrs by fluorescence assay | Homo sapiens | 1 | ALA4308881 | cell-based format | Scientific Literature | |
| 10. | ALA4334829 | B | Inhibition of human immunoproteasome beta 2i subunit at 10 uM using Boc-LRR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
| 11. | ALA4334851 | B | Inhibition of human immunoproteasome beta 2i subunit using Boc-LRR-AMC as substrate preincubated for 30 mins followed by substrate addition measured for 120 mins by fluorescence based assay | Homo sapiens | 10 | ALA4334435 | single protein format | Scientific Literature | |
| 12. | ALA4370444 | B | Inhibition of 20S immunoproteasome beta 2 (unknown origin) by cell based ABPP assay | Homo sapiens | 50 | ALA4368918 | cell-based format | Scientific Literature | |
| 13. | ALA4370448 | B | Inhibition of 20S immunoproteasome beta 2 in human Raji cell lysates after 1 hr by competitive ABPP assay | Homo sapiens | 17 | ALA4368918 | subcellular format | Scientific Literature | |
| 14. | ALA4370462 | B | Inhibition of 20S immunoproteasome beta 2 in human RPMI8226 cell lysates after 1 hr by coomassie brilliant blue staining-based fluorescence assay | Homo sapiens | 9 | ALA4368918 | subcellular format | Scientific Literature | |
| 15. | ALA4370468 | B | Inhibition of Morp-Ala-Tyr(O-C2H4-BODIPY(FL))-1-DecAla-EK binding to 20S immunoproteasome beta 2 in human Raji cell lysates at 0.3 uM in presence of 3-probe mixture by competitive ABPP assay | Homo sapiens | 1 | ALA4368918 | subcellular format | Scientific Literature | |
| 16. | ALA4370469 | B | Inhibition of Morp-Ala-Tyr(O-C2H4-BODIPY(FL))-1-DecAla-EK binding to 20S immunoproteasome beta 2 in human Raji cell lysates at 3 uM in presence of 3-probe mixture by competitive ABPP assay | Homo sapiens | 1 | ALA4368918 | subcellular format | Scientific Literature | |
| 17. | ALA4370471 | B | Inhibition of Morp-Ala-Tyr(O-C2H4-BODIPY(FL))-1-DecAla-EK binding to 20S immunoproteasome beta 2 in human Raji cell lysates at 1 uM in presence of 3-probe mixture by competitive ABPP assay | Homo sapiens | 1 | ALA4368918 | subcellular format | Scientific Literature | |
| 18. | ALA4370472 | B | Inhibition of 20S immunoproteasome beta 2 in intact human RPMI8226 cells after 1 hr by competitive ABPP assay | Homo sapiens | 2 | ALA4368918 | assay format | Scientific Literature | |
| 19. | ALA4370474 | B | Binding affinity to 20S immunoproteasome beta 2 in human Raji cell lysates at 3 uM by ABPP assay | Homo sapiens | 1 | ALA4368918 | subcellular format | Scientific Literature | |
| 20. | ALA4370475 | B | Inhibition of Morp-Ala-Tyr(O-C2H4-BODIPY(FL))-1-DecAla-EK binding to immunoproteasome beta 2 in human Raji cell lysates at 3 uM by competitive ABPP assay | Homo sapiens | 1 | ALA4368918 | subcellular format | Scientific Literature |
The page will load shortly, Thanks for your patience!