| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3418524 | B | Inhibition of TSSK3 (unknown origin) | Homo sapiens | 1 | ALA3414497 | single protein format | Scientific Literature | |
| 2. | ALA3631611 | B | Inhibition of TSSK3 (unknown origin) at 10 uM after 120 mins P33 radiolabeled kinase activity assay | Homo sapiens | 3 | ALA3627608 | single protein format | Scientific Literature | |
| 3. | ALA3750192 | B | Inhibition of human TSSK3 using [KKKVSRSGLYRSPSMPENLNRPR] as substrate | Homo sapiens | 1 | ALA3745707 | single protein format | Scientific Literature | |
| 4. | ALA3865681 | B | Inhibition of TSSK3 (unknown origin) | Homo sapiens | 1 | ALA3864189 | single protein format | Scientific Literature | |
| 5. | ALA4025424 | B | Inhibition of wild-type human full length TSSK3 (M1 to T268 residues) expressed in mammalian expression system assessed as residual activity at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4024706 | assay format | Scientific Literature | |
| 6. | ALA4044235 | B | Inhibition of wild-type human full length TSSK3 (M1 to T268 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control | Homo sapiens | 1 | ALA4043093 | cell-based format | Scientific Literature | |
| 7. | ALA4157314 | B | Binding affinity to wild-type human full length TSSK3 (M1 to T268 residues) expressed in mammalian expression system assessed as residual binding at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4152344 | assay format | Scientific Literature | |
| 8. | ALA4186093 | B | Binding affinity to wild-type human full length TSSK3 (M1 to T268 residues) expressed in HEK293 cells at 1 uM by Kinomescan method relative to control | Homo sapiens | 2 | ALA4184148 | cell-based format | Scientific Literature | |
| 9. | ALA4191221 | B | Inhibition of recombinant full-length human TSSK3 at 1 uM using AMARAASAAALARRR as substrate after 40 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4190187 | single protein format | Scientific Literature | |
| 10. | ALA4230993 | B | Binding affinity to wild-type human full length TSSK3 (M1 to T268 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4229344 | assay format | Scientific Literature | |
| 11. | ALA4264582 | B | Binding affinity to wild-type human full length TSSK3 (M1 to T268 residues) expressed in mammalian expression system assessed as remaining unbound target protein level at 1000 nM by Kinomescan method relative to control | Homo sapiens | 1 | ALA4261600 | assay format | Scientific Literature | |
| 12. | ALA4314633 | B | Inhibition of recombinant full-length human TSSK3 assessed as residual activity at 10 uM using AMARAASAAALARRR as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4311992 | single protein format | Scientific Literature | |
| 13. | ALA4322864 | B | Binding affinity to recombinant full-length N-terminal His-FLAG-GST-tagged TSSK3 (unknown origin) expressed in baculovirus infected Sf9 insect cells incubated for 1 hr by TR-FRET assay | Homo sapiens | 2 | ALA4321812 | cell-based format | Scientific Literature | |
| 14. | ALA4327913 | B | Inhibition of human TSSK3 assessed as residual activity at 1 uM using KKKVSRSGLYRSPSMPENLNRPR as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 2 | ALA4325871 | single protein format | Scientific Literature | |
| 15. | ALA4328277 | B | Inhibition of human TSSK3 assessed as residual activity at 100 uM using KKKVSRSGLYRSPSMPENLNRPR as substrate by [gamma-33P]-ATP assay relative to control | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
| 16. | ALA4328641 | B | Inhibition of human TSSK3 using KKKVSRSGLYRSPSMPENLNRPR as substrate by [gamma-33P]-ATP assay | Homo sapiens | 1 | ALA4325871 | single protein format | Scientific Literature | |
| 17. | ALA4335327 | B | Inhibition of recombinant full-length human TSSK3 at 1 uM assessed as residual activity at 1 uM using AMARAASAAALARRR as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method relative to control | Homo sapiens | 2 | ALA4334438 | single protein format | Scientific Literature | |
| 18. | ALA4337151 | B | Inhibition of recombinant full-length human TSSK3 assessed as residual activity at 10 uM using AMARAASAAALARRR as substrate incubated for 40 mins in presence of [gamma33P]ATP by scintillation counting based radiometry assay relative to control | Homo sapiens | 1 | ALA4334471 | single protein format | Scientific Literature | |
| 19. | ALA4352099 | B | Inhibition of recombinant full-length human TSSK3 at 10 uM using AMARAASAAALARRR as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA4350961 | single protein format | Scientific Literature | |
| 20. | ALA4352576 | B | Inhibition of human TSSK3 at 10 uM using KKKVSRSGLYRSPSMPENLNRPR as substrate in presence of [gamma-33P]-ATP | Homo sapiens | 1 | ALA4350963 | single protein format | Scientific Literature |
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