# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA860902 | B | Average Binding Constant for CSNK1E; NA=Not Active at 10 uM | Homo sapiens | 20 | ALA1144455 | single protein format | Scientific Literature | |
2. | ALA937637 | B | Inhibition of CK1epsilon | 1 | ALA1145498 | single protein format | Scientific Literature | ||
3. | ALA1025754 | B | Binding affinity to human CK1e at 10 uM relative to control | Homo sapiens | 17 | ALA1151712 | single protein format | Scientific Literature | |
4. | ALA1033258 | B | Inhibition of CSNK1E at 3 uM | 1 | ALA1142492 | single protein format | Scientific Literature | ||
5. | ALA1054858 | B | Inhibition of CK1epsilon at 10 uM by HotSpot assay relative to control | 1 | ALA1153464 | single protein format | Scientific Literature | ||
6. | ALA1050834 | B | Binding constant for full-length CSNK1E | Homo sapiens | 38 | ALA1150977 | single protein format | Scientific Literature | |
7. | ALA1052902 | B | Inhibition of CSNK1E assessed as enzyme activity at 1 uM relative to untreated control | 1 | ALA1155237 | single protein format | Scientific Literature | ||
8. | ALA1039038 | B | Binding affinity to CSNK1E assessed as dissociation constant | 1 | ALA1156118 | single protein format | Scientific Literature | ||
9. | ALA1045467 | B | Inhibition of recombinant CK1epsilon by Cherenkov counting in presence of 20 uM ATP | 2 | ALA1155278 | single protein format | Scientific Literature | ||
10. | ALA1066645 | B | Residual activity of CK1epsilon at 0.1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
11. | ALA1037107 | B | Residual activity of CK1epsilon at 1 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
12. | ALA1044275 | B | Residual activity of CK1epsilon at 10 uM by microplate scintillation counting | 3 | ALA1152560 | single protein format | Scientific Literature | ||
13. | ALA1102782 | B | Inhibition of CSNK1E at 10 uM | 2 | ALA1154277 | single protein format | Scientific Literature | ||
14. | ALA1114859 | B | Inhibition of CK1epsilon at 5 uM | 1 | ALA1154316 | single protein format | Scientific Literature | ||
15. | ALA1111813 | B | Binding affinity to CSNK1epsilon | 1 | ALA1156258 | single protein format | Scientific Literature | ||
16. | ALA1168840 | B | Inhibition of CSNK1E at 1 uM | 10 | ALA1165965 | single protein format | Scientific Literature | ||
17. | ALA1174186 | B | Inhibition of CSNK1E at 10 uM | 2 | ALA1177794 | single protein format | Scientific Literature | ||
18. | ALA1244400 | B | Inhibition of CK1epsilon at 1 uM after 60 mins by FRET assay in presence of 10 uM ATP | 7 | ALA1240340 | single protein format | Scientific Literature | ||
19. | ALA1244778 | B | Binding affinity to CSNK1E | 7 | ALA1240346 | single protein format | Scientific Literature | ||
20. | ALA1252288 | B | Inhibition of CSNK1E at 1 uM in presence of 10 uM ATP by Select Screen kinase assay relative to untreated control | 3 | ALA1250448 | single protein format | Scientific Literature |