# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA860902 | B | Average Binding Constant for CSNK1E; NA=Not Active at 10 uM | Homo sapiens | 20 | single protein format | Scientific Literature | ||
2. | ALA2091534 | B | Inhibition of CK1epsilon | 2 | single protein format | Scientific Literature | |||
3. | ALA1828475 | B | Inhibition of human CKI epsilon activity using Ser/Thr 11 peptide as substrate by FRET assay | Homo sapiens | 5 | single protein format | Scientific Literature | ||
4. | ALA1828205 | B | Activity of CSNK1E kinase at 1 uM | 1 | single protein format | Scientific Literature | |||
5. | ALA2066816 | B | Inhibition of human recombinant CK1epsilon by FRET assay | Homo sapiens | 11 | single protein format | Scientific Literature | ||
6. | ALA1908544 | B | Binding constant for CSNK1E kinase domain | 72 | single protein format | Scientific Literature | |||
7. | ALA1941719 | B | Inhibition of CK1epsilon at 10 uM by colorimetric analysis | 4 | single protein format | Scientific Literature | |||
8. | ALA1954390 | B | Inhibition of human CK1epsilon expressed in Escherichia coli BL21 using PLSRTLpSVASLPGL as substrate after 3 hrs by KinaseGlo assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
9. | ALA1958836 | B | Inhibition of CSNK1E at 1 uM | 1 | single protein format | Scientific Literature | |||
10. | ALA2014907 | B | Inhibition of CK1e at 10 uM | 1 | single protein format | Scientific Literature | |||
11. | ALA937637 | B | Inhibition of CK1epsilon | 1 | single protein format | Scientific Literature | |||
12. | ALA1025754 | B | Binding affinity to human CK1e at 10 uM relative to control | Homo sapiens | 17 | single protein format | Scientific Literature | ||
13. | ALA1033258 | B | Inhibition of CSNK1E at 3 uM | 1 | single protein format | Scientific Literature | |||
14. | ALA1054858 | B | Inhibition of CK1epsilon at 10 uM by HotSpot assay relative to control | 1 | single protein format | Scientific Literature | |||
15. | ALA1050834 | B | Binding constant for full-length CSNK1E | Homo sapiens | 38 | single protein format | Scientific Literature | ||
16. | ALA1052902 | B | Inhibition of CSNK1E assessed as enzyme activity at 1 uM relative to untreated control | 1 | single protein format | Scientific Literature | |||
17. | ALA1039038 | B | Binding affinity to CSNK1E assessed as dissociation constant | 1 | single protein format | Scientific Literature | |||
18. | ALA1045467 | B | Inhibition of recombinant CK1epsilon by Cherenkov counting in presence of 20 uM ATP | 2 | single protein format | Scientific Literature | |||
19. | ALA1066645 | B | Residual activity of CK1epsilon at 0.1 uM by microplate scintillation counting | 3 | single protein format | Scientific Literature | |||
20. | ALA1037107 | B | Residual activity of CK1epsilon at 1 uM by microplate scintillation counting | 3 | single protein format | Scientific Literature |